SCHEMBL11237837

SCHEMBL11237837

COc1ccc2c(c1)C(=O)C(CC#N)CC2

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.61
METAP1 P53582 3/20 0.51
CYP24A1 Q07973 6/20 0.49
CYP27A1 Q02318 3/20 0.49
CYP26A1 O43174 3/20 0.49
ACHE P22303 1/20 0.49
MTNR1A P48039 2/20 0.43
NQO2 P16083 1/20 0.42
MTNR1B P49286 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10341545 0.90 CYP24A1 (0.61) CYP19A1METAP1CYP24A1CYP27A1CYP26A1
SCHEMBL11011369 0.81 METAP1 (0.76) CYP19A1METAP1CYP24A1CYP27A1CYP26A1
SCHEMBL11239357 0.81 ACHE (0.47) ACHE
SCHEMBL9629597 0.81 MTNR1A (0.56) MTNR1ANQO2MTNR1B
SCHEMBL31028061 0.81 MTNR1A (0.56) MTNR1ANQO2MTNR1B
Hydrochloric Acid SCHEMBL4623159 0.80 METAP1 (0.78) CYP19A1METAP1CYP24A1CYP27A1CYP26A1
SCHEMBL8599809 0.80 CYP19A1 (0.62) CYP19A1METAP1CYP24A1CYP27A1CYP26A1
SCHEMBL8028175 0.79 CYP19A1 (0.61) CYP19A1METAP1CYP24A1CYP27A1CYP26A1
SCHEMBL9430945 0.79 CYP19A1 (0.61) CYP19A1METAP1CYP24A1CYP27A1CYP26A1
Iodide SCHEMBL9133365 0.79 CYP19A1 (0.61) CYP19A1METAP1CYP24A1CYP27A1CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309345-A POTASSIUM-SPARING DIURETICS CIBA-GEIGY CORPORATION (US) 1982-01-05 US disclosed
US-4173633-A DIURETICS CIBA-GEIGY CORPORATION (US) 1979-11-06 US disclosed