SCHEMBL11240576

SCHEMBL11240576

CC(C)C(C)(C)[SiH2]OC[C@H](C)[C@H]1CC[C@H]2[C@@H]3CC[C@H]4C(C(=O)c5ccccc5)C(=O)CC[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.45
SRD5A2 P31213 2/20 0.42
FNTA P49354 2/20 0.40
FNTB P49356 2/20 0.40
AKR1B10 O60218 1/20 0.40
AKR1B1 P15121 1/20 0.40
EFNA1 P20827 1/20 0.40
EPHA2 P29317 1/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPC1L1 Q9UHC9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11248546 0.85 SRD5A2 (0.43) GPBAR1SRD5A2FNTAFNTBNPC1L1
SCHEMBL11240580 0.85 SRD5A2 (0.43) GPBAR1SRD5A2FNTAFNTBNPC1L1
SCHEMBL11243498 0.84 SRD5A2 (0.59) GPBAR1SRD5A2FNTAFNTBAKR1B10
SCHEMBL11243490 0.84 SRD5A2 (0.59) GPBAR1SRD5A2FNTAFNTBAKR1B10
SCHEMBL11242975 0.78 CYP17A1 (0.50) GPBAR1SRD5A2FNTAFNTBACHE
SCHEMBL11242981 0.78 CYP17A1 (0.50) GPBAR1SRD5A2FNTAFNTBACHE
SCHEMBL11253127 0.76 SRD5A1 (0.39) SRD5A2ACHESRD5A1
SCHEMBL11253131 0.76 SRD5A1 (0.39) SRD5A2ACHESRD5A1
SCHEMBL11235256 0.75 CYP19A1 (0.51) GPBAR1SRD5A2LMNAKMT2AHSD17B10
SCHEMBL11235253 0.75 CYP19A1 (0.51) GPBAR1SRD5A2LMNAKMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4317817-A SKIN DISORDERS; ACEME; ENZYME INHIBITORS RICHARDSON-MERRELL INC. (US) 1982-03-02 US disclosed