SCHEMBL11240585

SCHEMBL11240585

CCCCCCc1[nH]c(=O)c(NC(C)=O)cc1-c1ccccn1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
APLNR P35414 1/20 0.38
JAK1 P23458 2/20 0.38
TYK2 P29597 2/20 0.38
ALOX12 P18054 1/20 0.38
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11239141 0.87 APLNR (0.40) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL11239131 0.82 APLNR (0.43) APLNR
SCHEMBL11248206 0.81 BTK (0.41) KDM4EALDH1A1HPGDHSD17B10APLNR
SCHEMBL11245687 0.81 PDE3B (0.49) KDM4EALDH1A1HPGDAPLNR
SCHEMBL11236502 0.80 PTGES (0.41) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL11239237 0.80 PARP1 (0.40) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL11232487 0.79 JAK1 (0.46) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL11238815 0.78 CDK5 (0.44) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL11230321 0.78 PDE3B (0.54) KDM4EALDH1A1HPGDAPLNR
SCHEMBL11239293 0.77 PDE3B (0.50) KDM4EALDH1A1HPGDAPLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed