SCHEMBL11240748

SCHEMBL11240748

C#Cc1cccc(OC(C)=O)c1.C1CC2CCC12

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FABP7 O15540 1/20 0.49
FABP5 Q01469 1/20 0.49
CYP3A4 P08684 1/20 0.49
LMNA P02545 1/20 0.49
ACHE P22303 1/20 0.45
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HTT P42858 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HAO1 Q9UJM8 1/20 0.40
MGLL Q99685 2/20 0.40
EPHX2 P34913 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3828627 0.91 LMNA (0.58) FABP7FABP5CYP3A4LMNAACHE
SCHEMBL11240283 0.80 HTR2C (0.45) CYP3A4ACHEALDH1A1
SCHEMBL26036690 0.77 FABP7 (0.49) FABP7FABP5CYP3A4LMNAACHE
SCHEMBL7679108 0.76 LMNA (0.59) CYP3A4LMNAACHEKMT2AMEN1
SCHEMBL16953007 0.74 LMNA (0.58) CYP3A4LMNAACHEKMT2AMEN1
SCHEMBL30676498 0.74 CYP3A4 (0.58) CYP3A4LMNAACHEKMT2AMEN1
SCHEMBL10547627 0.74 CYP3A4 (0.58) CYP3A4LMNAACHEKMT2AMEN1
SCHEMBL28036637 0.74 MEN1 (0.66) FABP7FABP5CYP3A4LMNAKMT2A
SCHEMBL11238391 0.73 EGFR (0.54) KMT2AMEN1ALDH1A1HSD17B10POLB
SCHEMBL11232887 0.73 LMNA (0.36) FABP7FABP5LMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4157449-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1979-06-05 US claimed
US-4365093-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1982-12-21 US disclosed
US-4296264-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1981-10-20 US disclosed
US-4288457-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1981-09-08 US disclosed
US-4264627-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1981-04-28 US disclosed
US-4171373-A Ethynylbenzene compounds and derivatives thereof to treat pain, fever and inflammation WILLIAM H. RORER, INC. (US) 1979-10-16 US disclosed
US-4168320-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1979-09-18 US disclosed
US-4166133-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF TO TREAT PAIN, FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1979-08-28 US disclosed
US-4157449-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1979-06-05 US disclosed
US-4150148-A NITROSUBSTITUTED WILLIAM H. RORER, INC. (US) 1979-04-17 US disclosed
US-4120889-A Cyano ethynylbenzene compounds WILLIAM H. RORER, INC. (US) 1978-10-17 US disclosed
US-4120885-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1978-10-17 US disclosed
US-4105786-A ANTIINFLAMMATORY WILLIAM H. RORER, INC. (US) 1978-08-08 US disclosed
US-4101591-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1978-07-18 US disclosed
US-4096279-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain fever and inflammation WILLIAM H. RORER, INC. (US) 1978-06-20 US disclosed
US-4094995-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF TO TREAT PAIN, FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1978-06-13 US disclosed
US-4093737-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain, fever or inflammation WILLIAM H. RORER, INC. (US) 1978-06-06 US disclosed
US-4075354-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF FOR TREATING PAIN FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1978-02-21 US disclosed
US-3981932-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1976-09-21 US disclosed