SCHEMBL1124170

SCHEMBL1124170

Cc1ccc(C=CC(=O)NCc2ccc(N3CCOCC3)nc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.62
KDM4E B2RXH2 1/20 0.53
MAPT P10636 5/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C19 P33261 1/20 0.50
LMNA P02545 7/20 0.49
KMT2A Q03164 4/20 0.49
MAPK1 P28482 1/20 0.49
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
ALDH1A1 P00352 4/20 0.48
PARP1 P09874 1/20 0.48
AOC3 Q16853 1/20 0.47
GAA P10253 3/20 0.46
HPGD P15428 2/20 0.46
TP53 P04637 1/20 0.46
THRB P10828 1/20 0.46
MEN1 O00255 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1124204 0.87 SMN1; SMN2 (0.53) SMN1; SMN2MAPTLMNAKMT2AMAPK1
SCHEMBL1124113 0.80 PARP1 (0.54) KDM4EMAPTCYP1A2CYP2C19CYP11B1
SCHEMBL3784304 0.74 ALDH1A1 (0.49) SMN1; SMN2KDM4EMAPTCYP1A2CYP2C19
SCHEMBL3784306 0.74 ALDH1A1 (0.49) SMN1; SMN2KDM4EMAPTCYP1A2CYP2C19
SCHEMBL1124168 0.74 AOC3 (0.50) SMN1; SMN2KDM4EMAPTCYP1A2CYP2C19
SCHEMBL1124174 0.74 AOC3 (0.50) SMN1; SMN2KDM4EMAPTCYP1A2CYP2C19
SCHEMBL29551688 0.74 PIM2 (0.54) SMN1; SMN2KDM4EMAPTCYP1A2CYP2C19
SCHEMBL3786488 0.74 PIM2 (0.54) SMN1; SMN2KDM4EMAPTCYP1A2CYP2C19
SCHEMBL3786486 0.74 PIM2 (0.54) SMN1; SMN2KDM4EMAPTCYP1A2CYP2C19
SCHEMBL14303030 0.74 ALDH1A1 (0.40) SMN1; SMN2KDM4EMAPTLMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282996-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS Actelion Pharmaceuticals Ltd. (CH) 2011-02-16 EP claimed
EP-2282996-A1 TETRAHYDROISOQUINOLINES AS ANTIMALARIAL AGENTS Actelion Pharmaceuticals Ltd. (CH) 2011-02-16 EP disclosed