SCHEMBL11242151

SCHEMBL11242151

CN1C(=O)CCc2c(OCCCNCCCO)cccc21

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 1/20 0.44
TSHR P16473 2/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HTR6 P50406 5/20 0.40
ALDH1A1 P00352 2/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
PTPN1 P18031 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11237380 0.99 DRD3 (0.43) DRD3TSHRTP53CYP1A2CYP3A4
SCHEMBL11367098 0.87 HTR6 (0.44) DRD3TSHRTP53CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11234315 0.87 HTR6 (0.40) DRD3HTR6L3MBTL1HRH3PTPN1
Hydrochloric Acid SCHEMBL11231511 0.86 HTR6 (0.43) DRD3TSHRTP53CYP1A2CYP3A4
SCHEMBL11227272 0.86 KDM4E (0.38) DRD3TDP1HTR6ALDH1A1HRH3
SCHEMBL11362472 0.81 HTR6 (0.41) DRD3TSHRTP53CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11250180 0.81 HTR6 (0.60) TSHRTP53CYP1A2CYP3A4CYP2D6
SCHEMBL9653138 0.79 HRH3 (0.40) HTR6HRH3
SCHEMBL11724685 0.75 CYP1A2 (0.46) TSHRCYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL11386590 0.74 HTR6 (0.41) TDP1HTR6ALDH1A1HRH3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4256890-A ADRENERGIC BLOCKING AGENTS OTSUKAPHARMACEUTICAL CO., LTD. (JP) 1981-03-17 US claimed
US-4329468-A ADRENERGIC BLOCKING AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1982-05-11 US disclosed
US-4256890-A ADRENERGIC BLOCKING AGENTS OTSUKAPHARMACEUTICAL CO., LTD. (JP) 1981-03-17 US disclosed