SCHEMBL11242404

SCHEMBL11242404

COC(=O)CCCOc1ccc(CC(C)NCC(O)c2ccccc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 14/20 0.61
ADRB1 P08588 11/20 0.61
ADRB2 P07550 10/20 0.61
GLA P06280 1/20 0.61
SLC2A1 P11166 2/20 0.59
CYP2D6 P10635 2/20 0.57
ADRA1D P25100 1/20 0.57
ADRA1A P35348 1/20 0.57
ADRA1B P35368 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
CYP3A4 P08684 1/20 0.52
HIF1A Q16665 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11247530 0.88 ADRB3 (0.77) ADRB3ADRB1ADRB2GLASLC2A1
SCHEMBL11251142 0.88 ADRB3 (0.77) ADRB3ADRB1ADRB2GLASLC2A1
SCHEMBL10933710 0.85 ADRB2 (0.60) ADRB3ADRB1ADRB2GLASLC2A1
SCHEMBL7150585 0.84 ADRB3 (0.77) ADRB3ADRB1ADRB2GLASLC2A1
SCHEMBL7150582 0.84 ADRB3 (0.77) ADRB3ADRB1ADRB2GLASLC2A1
Bromide SCHEMBL11148850 0.83 ADRB2 (0.60) ADRB3ADRB1ADRB2GLASLC2A1
SCHEMBL10478199 0.83 ADRB3 (0.78) ADRB3ADRB1ADRB2GLASLC2A1
SCHEMBL10913821 0.82 ADRB2 (0.49) ADRB3ADRB1ADRB2GLASLC2A1
Hydrochloric Acid SCHEMBL10935778 0.82 SLC2A1 (0.56) ADRB3ADRB1ADRB2GLASLC2A1
SCHEMBL11255869 0.82 ADRB3 (0.77) ADRB3ADRB1ADRB2GLASLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US claimed
EP-0023385-B1 ETHANAMINE DERIVATIVES, THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS BEECHAM GROUP PLC (GB) 1982-12-15 EP disclosed
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US disclosed
EP-0023385-A1 Ethanamine derivatives, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-02-04 EP disclosed