SCHEMBL11247530

SCHEMBL11247530

COC(=O)COc1ccc(CC(C)NCC(O)c2ccccc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 15/20 0.77
ADRB1 P08588 13/20 0.77
ADRB2 P07550 12/20 0.77
GLA P06280 1/20 0.77
CYP2D6 P10635 2/20 0.66
ADRA1D P25100 1/20 0.66
ADRA1A P35348 1/20 0.66
ADRA1B P35368 1/20 0.66
CYP1A2 P05177 1/20 0.66
CYP2C9 P11712 1/20 0.66
CYP2C19 P33261 1/20 0.66
CYP3A4 P08684 1/20 0.60
HIF1A Q16665 1/20 0.60
SLC2A1 P11166 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11251142 1.00 ADRB3 (0.77) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL10478199 0.91 ADRB3 (0.78) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL11255869 0.89 ADRB3 (0.77) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL11246376 0.89 ADRB3 (0.62) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL11253857 0.88 ADRB3 (0.77) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL11242404 0.88 ADRB3 (0.61) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL10859889 0.87 ADRB3 (0.63) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL11255890 0.87 ADRB3 (0.77) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL11245796 0.87 ADRB3 (0.65) ADRB3ADRB1ADRB2GLACYP2D6
SCHEMBL5144151 0.87 ADRB3 (1.00) ADRB3ADRB1ADRB2GLACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US claimed
EP-0023385-B1 ETHANAMINE DERIVATIVES, THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS BEECHAM GROUP PLC (GB) 1982-12-15 EP disclosed
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US disclosed
EP-0023385-A1 Ethanamine derivatives, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-02-04 EP disclosed