SCHEMBL11243333

SCHEMBL11243333

Cn1nc(-c2ccncc2)cc(C(=O)NN)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 1/20 0.42
CLK1 P49759 1/20 0.42
UBE2N P61088 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CASP1 P29466 3/20 0.42
MPO P05164 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C19 P33261 1/20 0.41
GPR142 Q7Z601 2/20 0.41
MAPK13 O15264 2/20 0.41
MAPK12 P53778 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11247419 0.85 KDM4E (0.44) KDM4ERAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL11245225 0.85 CASP1 (0.51) ALDH1A1HPGDMAPK1CLK1UBE2N
SCHEMBL11242637 0.84 KDM4E (0.46) KDM4ERAB9ASMN1; SMN2ALDH1A1HPGD
Ammonia Solution, Strong SCHEMBL11371806 0.83 CASP1 (0.50) ALDH1A1HPGDMAPK1CLK1UBE2N
SCHEMBL11241157 0.83 KDM4E (0.43) KDM4ERAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL11248350 0.83 KDM4E (0.45) KDM4ERAB9ASMN1; SMN2ALDH1A1CASP1
SCHEMBL11235913 0.83 DHODH (0.46) KDM4ESMN1; SMN2ALDH1A1HPGDMAPK1
SCHEMBL11246089 0.81 KDM4E (0.41) KDM4ERAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL11241921 0.81 KDM4E (0.44) KDM4ERAB9ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL11231677 0.81 CNR1 (0.43) KDM4ERAB9ASMN1; SMN2MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4346221-A Preparation of 4-amino-6-(pyridinyl)-3(2H)-pyridazinones from 6-(pyridinyl)-3(2H)-pyridazinones STERLING DRUG INC. (US) 1982-08-24 US disclosed
US-4338446-A Di-(lower-alkyl)hydroxy-[2-oxo-2-(pyridinyl)ethyl]-propanedioates STERLING DRUG INC. (US) 1982-07-06 US disclosed
US-4305943-A 4-Amino-6-(pyridinyl)-3(2H)-pyridazinones and their use as cardiotonics STERLING DRUG INC. (US) 1981-12-15 US disclosed
US-4304776-A 4-Substituted-6-(pyridinyl)-3(2h)-pyridazinones and their use as intermediates and cardiotonics STERLING DRUG INC. (US) 1981-12-08 US disclosed