SCHEMBL11235913

SCHEMBL11235913

Cn1nc(-c2ccncc2)cc(C(=O)O)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.46
ALDH1A1 P00352 3/20 0.45
GAA P10253 1/20 0.45
GSK3B P49841 8/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
MAPK1 P28482 1/20 0.43
CLK1 P49759 1/20 0.43
UBE2N P61088 1/20 0.43
GPR142 Q7Z601 1/20 0.41
HTT P42858 1/20 0.41
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CASP1 P29466 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPK14 Q16539 1/20 0.39
CDC7 O00311 1/20 0.39
ROCK2 O75116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11245225 0.87 CASP1 (0.51) ALDH1A1HPGDHSD17B10MAPK1CLK1
Ammonia Solution, Strong SCHEMBL11371806 0.85 CASP1 (0.50) ALDH1A1HPGDHSD17B10MAPK1CLK1
SCHEMBL11243333 0.83 KDM4E (0.47) ALDH1A1GSK3BHPGDHSD17B10MAPK1
SCHEMBL11239782 0.82 GSK3B (0.41) DHODHALDH1A1GAAGSK3BHPGD
SCHEMBL11240735 0.81 DHODH (0.43) DHODHALDH1A1GAAGSK3BHPGD
SCHEMBL11230958 0.81 PDE4B (0.43) DHODHALDH1A1GAAGSK3BHPGD
SCHEMBL11236330 0.81 ALDH1A1 (0.63) ALDH1A1GAAGSK3BHPGDHSD17B10
SCHEMBL11233660 0.80 DHODH (0.42) DHODHALDH1A1GAAGSK3BHPGD
SCHEMBL7275259 0.80 PHGDH (0.48) ALDH1A1GAAHPGDKDM4ECASP1
SCHEMBL30722885 0.80 PTPN1 (0.50) GSK3BGPR142KDM4ECDC7ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4346221-A Preparation of 4-amino-6-(pyridinyl)-3(2H)-pyridazinones from 6-(pyridinyl)-3(2H)-pyridazinones STERLING DRUG INC. (US) 1982-08-24 US disclosed
US-4338446-A Di-(lower-alkyl)hydroxy-[2-oxo-2-(pyridinyl)ethyl]-propanedioates STERLING DRUG INC. (US) 1982-07-06 US disclosed
US-4305943-A 4-Amino-6-(pyridinyl)-3(2H)-pyridazinones and their use as cardiotonics STERLING DRUG INC. (US) 1981-12-15 US disclosed
US-4304776-A 4-Substituted-6-(pyridinyl)-3(2h)-pyridazinones and their use as intermediates and cardiotonics STERLING DRUG INC. (US) 1981-12-08 US disclosed