SCHEMBL11243532

SCHEMBL11243532

CCCc1ncc(N)cc1-c1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 5/20 0.38
IMPDH2 P12268 1/20 0.38
FYN P06241 1/20 0.38
PDE3B Q13370 3/20 0.37
PDE3A Q14432 3/20 0.37
CDC7 O00311 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
PIM1 P11309 1/20 0.36
PRKACA P17612 1/20 0.36
CDK2 P24941 1/20 0.36
GSK3B P49841 1/20 0.36
HIPK2 Q9H2X6 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
AURKB Q96GD4 2/20 0.36
INCENP Q9NQS7 2/20 0.36
AURKA O14965 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11240217 0.92 CYP3A4 (0.41) NTRK1IMPDH2FYNPDE3BPDE3A
SCHEMBL11244037 0.91 KDM4E (0.44) NTRK1IMPDH2FYNPDE3BPDE3A
SCHEMBL11238028 0.80 NTRK1 (0.37) NTRK1IMPDH2FYNPDE3BPDE3A
SCHEMBL11236122 0.75 FYN (0.45) NTRK1IMPDH2FYNPDE3BPDE3A
SCHEMBL4604967 0.72 KDM4E (0.35) KDM4EMEN1USP2ALDH1A1GAA
SCHEMBL11065116 0.71 GABRP (0.42) PDE3BPDE3AGSK3BCYP3A4CYP2D6
SCHEMBL11228166 0.71 NTRK1 (0.40) NTRK1IMPDH2FYNPDE3BPDE3A
SCHEMBL31165734 0.71 AURKA (0.59) NTRK1FYNGSK3BCYP3A4CYP2D6
SCHEMBL11236599 0.71 AURKB (0.41) NTRK1IMPDH2FYNPDE3BPDE3A
SCHEMBL30772309 0.69 PDE3B (0.40) FYNPDE3BPDE3ACYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309537-A Production of imidazo[4,5-b]pyridin-2-ones or thiones STERLING DRUG INC. (US) 1982-01-05 US disclosed
US-4297360-A 5-(Pyridinyl)pyridine-2,3-diamines, preparation thereof and their cardiotonic use STERLING DRUG INC. (US) 1981-10-27 US disclosed
US-4294837-A 1,3-Dihydro-6-(pyridinyl)-2H-imidazo[4,5-b]pyridin-2-ones and -imidazo[4,5-b]pyridine-2-thiones and their cardiotonic use STERLING DRUG INC. (US) 1981-10-13 US disclosed
US-4276293-A Compositions and their preparation STERLING DRUG INC. (US) 1981-06-30 US disclosed