SCHEMBL11244112

SCHEMBL11244112

CC1(C)COC(CCCCn2ccnc2)(c2ccc(Cl)cc2)OC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.47
ALDH1A1 P00352 1/20 0.47
QPCT Q16769 2/20 0.45
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
HMOX1 P09601 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
CYP2B6 P20813 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11242901 0.97 QPCT (0.46) TP53ALDH1A1QPCTKDM4ETSHR
SCHEMBL11240587 0.92 TP53 (0.44) TP53ALDH1A1QPCTKDM4ETSHR
SCHEMBL11242340 0.90 QPCT (0.47) TP53ALDH1A1QPCTTSHRCYP19A1
SCHEMBL11241853 0.88 CYP19A1 (0.44) CYP19A1CYP11B1CYP11B2
SCHEMBL11230058 0.88 TP53 (0.51) TP53ALDH1A1QPCTKDM4ETSHR
SCHEMBL11241810 0.87 MEN1 (0.52) TP53ALDH1A1QPCTKDM4ETSHR
SCHEMBL11241916 0.86 QPCT (0.48) TP53ALDH1A1QPCTKDM4ETSHR
SCHEMBL11242197 0.86 QPCT (0.49) TP53ALDH1A1QPCTKDM4ETSHR
SCHEMBL11245761 0.85 LMNA (0.43) QPCTKDM4ETSHRCYP19A1
SCHEMBL11233658 0.85 CYP19A1 (0.45) CYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0049565-A2 Derivatives of substituted N-alkylimidazoles, their preparation and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1982-04-14 EP disclosed
US-4321272-A Derivatives of substituted N-alkylimidazoles SYNTEX (U.S.A.) INC. (US) 1982-03-23 US disclosed