SCHEMBL11244642

SCHEMBL11244642

CCOC(=O)c1ccc2c(c1)nc(N)n2S(=O)(=O)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 1/20 0.48
ALDH1A1 P00352 5/20 0.47
HPGD P15428 3/20 0.47
SIRT2 Q8IXJ6 5/20 0.46
SIRT1 Q96EB6 4/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
PDE2A O00408 1/20 0.45
PTGER4 P35408 1/20 0.45
MAPT P10636 4/20 0.44
NLRP3 Q96P20 1/20 0.44
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.42
GAA P10253 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11258832 0.91 PI4KB (0.59) PI4KBALDH1A1NPC1RAB9AMEN1
SCHEMBL10643222 0.85 PI4KB (0.51) PI4KBKMT2ACYP3A4
SCHEMBL11152574 0.84 SIRT2 (0.48) ALDH1A1HPGDSIRT2SIRT1NPC1
SCHEMBL8253380 0.79 SIRT2 (0.52) ALDH1A1HPGDSIRT2SIRT1NPC1
SCHEMBL18058954 0.79 MAPK14 (0.47) PI4KBCYP3A4
SCHEMBL10643033 0.79 PI4KB (0.61) PI4KBALDH1A1HPGDMAPTKDM4E
SCHEMBL22382307 0.78 KMT2A (0.63) ALDH1A1HPGDSIRT2SIRT1NPC1
SCHEMBL18058988 0.78 PI4KB (0.49) PI4KBGAACYP3A4
SCHEMBL22382508 0.77 SIRT2 (0.51) ALDH1A1HPGDSIRT2SIRT1NPC1
SCHEMBL10640202 0.76 PI4KB (0.47) PI4KBMEN1KMT2AGAACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4316021-A VIRICIDES ELI LILLY AND COMPANY (US) 1982-02-16 US disclosed
US-4243813-A VIRICIDES ELI LILLY AND COMPANY (US) 1981-01-06 US disclosed
US-4196125-A VIRICIDES ELI LILLY AND COMPANY (US) 1980-04-01 US disclosed
US-4118573-A ANTIVIRAL AGENTS ELI LILLY AND COMPANY (US) 1978-10-03 US disclosed
US-4018790-A VIRICIDES ELI LILLY AND COMPANY (US) 1977-04-19 US disclosed