SCHEMBL11258832

SCHEMBL11258832

CCOC(=O)c1ccc2nc(N)n(S(=O)(=O)C(C)C)c2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 1/20 0.59
MAPK14 Q16539 14/20 0.47
CYP3A4 P08684 8/20 0.47
PDE2A O00408 1/20 0.45
ABL1 P00519 1/20 0.43
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
FYN P06241 1/20 0.43
PIM1 P11309 1/20 0.43
FGFR1 P11362 1/20 0.43
MAPK1 P28482 1/20 0.43
FLT4 P35916 1/20 0.43
KDR P35968 1/20 0.43
MAPK8 P45983 1/20 0.43
MAPK9 P45984 1/20 0.43
CSNK1D P48730 1/20 0.43
LIMK1 P53667 1/20 0.43
DYRK1A Q13627 1/20 0.43
CDC42BPA Q5VT25 1/20 0.43
AURKB Q96GD4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11244642 0.91 PI4KB (0.48) PI4KBCYP3A4PDE2AALDH1A1KDM4E
SCHEMBL11076745 0.85 PI4KB (0.62) PI4KBMAPK14CYP3A4ABL1EGFR
SCHEMBL11733042 0.84 PDE2A (0.45) PI4KBCYP3A4PDE2AALDH1A1KDM4E
SCHEMBL11151131 0.84 PDE2A (0.45) PI4KBMAPK14CYP3A4PDE2AALDH1A1
SCHEMBL11622008 0.84 PI4KB (0.59) PI4KBMAPK14CYP3A4ABL1EGFR
SCHEMBL11257304 0.83 PDE2A (0.44) PI4KBCYP3A4PDE2AALDH1A1KDM4E
SCHEMBL11148345 0.83 PI4KB (0.61) PI4KBMAPK14CYP3A4
SCHEMBL11148343 0.83 PI4KB (0.61) PI4KBMAPK14CYP3A4
SCHEMBL11622012 0.82 NOD1 (0.55) PI4KBPDE2AALDH1A1NPC1RAB9A
SCHEMBL11164281 0.82 PI4KB (0.60) PI4KBMAPK14CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4118573-A ANTIVIRAL AGENTS ELI LILLY AND COMPANY (US) 1978-10-03 US claimed
US-4316021-A VIRICIDES ELI LILLY AND COMPANY (US) 1982-02-16 US disclosed
US-4243813-A VIRICIDES ELI LILLY AND COMPANY (US) 1981-01-06 US disclosed
US-4196125-A VIRICIDES ELI LILLY AND COMPANY (US) 1980-04-01 US disclosed
US-4118573-A ANTIVIRAL AGENTS ELI LILLY AND COMPANY (US) 1978-10-03 US disclosed
US-4018790-A VIRICIDES ELI LILLY AND COMPANY (US) 1977-04-19 US disclosed