SCHEMBL11244775

SCHEMBL11244775

CN(C)Cc1cccc(OCCCN=C(NC#N)NCCCCCCCCCCCCNC(=NCCCOc2cccc(CN(C)C)c2)NC#N)c1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 4/20 0.42
HRH2 P25021 2/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11209515 0.97 BCHE (0.42) HRH4HRH2BCHEACHE
SCHEMBL9870811 0.89 ACHE (0.41) BCHEACHE
SCHEMBL9870816 0.89 ACHE (0.41) BCHEACHE
SCHEMBL9870818 0.86 HRH4 (0.44) HRH4
SCHEMBL11371367 0.83 ACHE (0.69) BCHEACHE
SCHEMBL11244766 0.83 ACHE (0.40) BCHEACHE
SCHEMBL11209512 0.81 CYP2D6 (0.40) BCHEACHE
SCHEMBL11290548 0.80 ACHE (0.42) BCHEACHE
SCHEMBL11290545 0.80 ACHE (0.42) BCHEACHE
SCHEMBL11374134 0.80 CYP2D6 (0.40) BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4366164-A HISTAMINE H2-ANTAGONISTS GLAXO GROUP LIMITED (GB) 1982-12-28 US disclosed
US-4317819-A Amine derivatives GLAXO GROUP LIMITED (GB) 1982-03-02 US disclosed
US-4264614-A HISTAMINE ANTAGONIST; ANTIALLERGENS; ANTISECRETORY AND ANTIINFLAMMATORY AGENTS GLAXO GROUP LIMITED (GB) 1981-04-28 US disclosed