SCHEMBL11245229

SCHEMBL11245229

COCCN=C(N)Nc1nc(-c2cccc(N(C)C(N)=NC#N)c2)cs1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 16/20 0.48
ATP4B P51164 16/20 0.48
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CASP3 P42574 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
EBP Q15125 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11252548 0.86 ATP4A (0.43) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL11245308 0.83 ABL1 (0.41) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL11245218 0.82 ATP4A (0.49) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL11245222 0.82 ATP4A (0.49) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL11245371 0.80 ATP4A (0.57) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL11245367 0.80 ATP4A (0.57) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL11254016 0.79 ATP4A (0.41) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL10673686 0.74 ABL1 (0.39) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL11260913 0.72 ATP4A (0.39) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL10976747 0.72 AOC3 (0.36) ATP4AATP4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4315009-A Antisecretory guanidine derivatives and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-02-09 US claimed
EP-0003640-B1 ANTISECRETORY GUANIDINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-01-27 EP claimed
EP-0003640-A2 Antisecretory guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-08-22 EP claimed
US-4315009-A Antisecretory guanidine derivatives and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-02-09 US disclosed
EP-0003640-B1 ANTISECRETORY GUANIDINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-01-27 EP disclosed
EP-0003640-A2 Antisecretory guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-08-22 EP disclosed