SCHEMBL11245367

SCHEMBL11245367

COCC/N=C(/N)Nc1nc(-c2cccc(N)c2)cs1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 9/20 0.57
ATP4B P51164 9/20 0.57
HDAC3 O15379 6/20 0.51
HDAC1 Q13547 6/20 0.51
HDAC2 Q92769 6/20 0.51
HDAC10 Q969S8 6/20 0.51
HDAC6 Q9UBN7 4/20 0.51
HDAC8 Q9BY41 3/20 0.51
HDAC4 P56524 2/20 0.51
HDAC7 Q8WUI4 2/20 0.51
HDAC11 Q96DB2 2/20 0.51
HDAC9 Q9UKV0 2/20 0.51
HDAC5 Q9UQL6 2/20 0.51
NCOR2 Q9Y618 1/20 0.48
TSHR P16473 1/20 0.46
RECQL P46063 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11245371 1.00 ATP4A (0.57) ATP4AATP4BHDAC3HDAC1HDAC2
SCHEMBL10751731 0.82 HDAC3 (0.56) ATP4AATP4BHDAC3HDAC1HDAC2
SCHEMBL10751726 0.82 HDAC3 (0.56) ATP4AATP4BHDAC3HDAC1HDAC2
SCHEMBL11245218 0.80 ATP4A (0.49) ATP4AATP4BHDAC3HDAC1HDAC2
SCHEMBL11245222 0.80 ATP4A (0.49) ATP4AATP4BHDAC3HDAC1HDAC2
Bromide SCHEMBL11247478 0.80 KMT2A (0.59) ATP4AATP4BNPC1RAB9AALDH1A1
Bromide SCHEMBL11247477 0.80 KMT2A (0.59) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL11245229 0.80 ATP4A (0.48) ATP4AATP4BNPC1RAB9AALDH1A1
SCHEMBL2393684 0.75 HDAC3 (0.59) HDAC3HDAC1HDAC2HDAC10HDAC6
SCHEMBL15689011 0.74 ABL1 (0.74) HDAC3HDAC1HDAC2HDAC10HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4315009-A Antisecretory guanidine derivatives and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-02-09 US disclosed
EP-0003640-B1 ANTISECRETORY GUANIDINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-01-27 EP disclosed
EP-0003640-A2 Antisecretory guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-08-22 EP disclosed