SCHEMBL11245665

SCHEMBL11245665

CSCC[C@@H](C(=O)O)N(Cc1ccccc1)C(=O)CCS

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
POLB P06746 1/20 0.41
HSD17B10 Q99714 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KDM4E B2RXH2 1/20 0.38
FNTA P49354 2/20 0.37
FNTB P49356 2/20 0.37
ACE P12821 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
ANPEP P15144 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11128323 0.81 KMT2A (0.45) KMT2AMEN1ALDH1A1LMNAPOLB
SCHEMBL11271369 0.81 MEN1 (0.52) KMT2AMEN1ALDH1A1LMNAPOLB
SCHEMBL11251274 0.81 KMT2A (0.44) KMT2AMEN1ALDH1A1LMNAPOLB
SCHEMBL11252020 0.79 KMT2A (0.42) KMT2AMEN1ALDH1A1LMNAPOLB
SCHEMBL6681598 0.78 ANPEP (0.42) KMT2AMEN1NPC1RAB9AFNTA
SCHEMBL27768608 0.78 ANPEP (0.42) KMT2AMEN1NPC1RAB9AFNTA
SCHEMBL11252386 0.78 KMT2A (0.49) KMT2AMEN1ALDH1A1LMNAPOLB
SCHEMBL9081277 0.77 NPC1 (0.42) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL2328144 0.76 MEN1 (0.45) KMT2AMEN1ALDH1A1LMNAPOLB
SCHEMBL9082541 0.75 LMNA (0.43) KMT2AMEN1ALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0066956-A1 Enkephalinase enzyme inhibiting compounds PFIZER INC. (US) 1982-12-15 EP disclosed
US-4329495-A USEFUL AS ANALGESICS OR ANTICONVULSANTS, CHIRAL 2-(2-BENZYL-3-MERCAPTOPROPIONYLAMINO)-THIOBUTYRIC ACIDS, OR ALKANOL DERIVATIVES PFIZER INC. (US) 1982-05-11 US disclosed