SCHEMBL11246290

SCHEMBL11246290

c1ccc(-c2ccccc2-c2nc3c4ccccc4ccn3n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.43
NPC1 O15118 3/20 0.42
RAB9A P51151 2/20 0.42
DHODH Q02127 1/20 0.40
PARP1 P09874 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.39
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
MAPK1 P28482 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
ATM Q13315 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11416817 0.87 DHODH (0.50) CYP11B2NPC1RAB9ADHODHPARP1
SCHEMBL11262382 0.84 DHODH (0.55) CYP11B2NPC1RAB9ADHODHPARP1
SCHEMBL11250627 0.81 DHODH (0.45) DHODHPARP1ADORA3ADORA1PDE10A
SCHEMBL21306416 0.79 PDE10A (0.48) CYP11B2NPC1RAB9ADHODHPARP1
SCHEMBL11600859 0.78 CYP1A2 (0.45) CYP11B2NPC1RAB9AKDM4EALDH1A1
Lotrifen SCHEMBL2107797 0.76 NR1H3 (0.47) CYP11B2NPC1RAB9ADHODHPARP1
SCHEMBL11413909 0.76 AHR (0.63) NPC1RAB9ADHODHPARP1KDM4E
SCHEMBL11407248 0.75 CYP11B2 (0.42) CYP11B2DHODHPARP1ABCG2KDM4E
SCHEMBL11419299 0.75 HSD17B2 (0.47) NPC1RAB9ADHODHPARP1ALDH1A1
SCHEMBL11407906 0.75 CYP11B2 (0.41) CYP11B2NPC1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4313950-A Antireproductive tricyclic ortho-fused nitrogen containing compounds GRUPPO LEPETIT S.P.A. (IT) 1982-02-02 US disclosed
US-4275066-A 1,2,4-TRIAZOLO(5.1A)ISOINDOZE, TRIAZOLO(5.1A) ISOQUINOLINE OR 1,2,4,-TRIAZOLO (5.1A)(2) BENZAZEPINE CONTRACEPTIVES GRUPPO LEPETIT S.P.A. (IT) 1981-06-23 US disclosed