SCHEMBL11262382

SCHEMBL11262382

c1ccc(-c2ccc(-c3nc4c5ccccc5ccn4n3)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.55
PARP1 P09874 1/20 0.48
AHR P35869 1/20 0.46
ADORA3 P0DMS8 4/20 0.45
ADORA1 P30542 2/20 0.45
PDE10A Q9Y233 2/20 0.43
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
GABRA4 P48169 1/20 0.41
GABRE P78334 1/20 0.41
GABRA6 Q16445 1/20 0.41
GABRG1 Q8N1C3 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11416817 0.97 DHODH (0.50) DHODHPARP1AHRADORA3ADORA1
SCHEMBL11250627 0.89 DHODH (0.45) DHODHPARP1AHRADORA3ADORA1
SCHEMBL21306416 0.88 PDE10A (0.48) DHODHPARP1AHRADORA3ADORA1
Lotrifen SCHEMBL2107797 0.88 NR1H3 (0.47) DHODHPARP1AHRADORA3ADORA1
SCHEMBL11413909 0.88 AHR (0.63) DHODHPARP1AHRADORA3KDR
SCHEMBL11246290 0.84 CYP11B2 (0.43) DHODHPARP1AHRADORA3ADORA1
SCHEMBL11417325 0.84 ADORA3 (0.46) DHODHAHRADORA3ADORA1GAA
SCHEMBL11241095 0.83 DHODH (0.48) DHODHPARP1AHRADORA3ADORA1
SCHEMBL11267545 0.83 DHODH (0.48) DHODHPARP1AHRADORA3ADORA1
SCHEMBL11413315 0.82 THRB (0.46) DHODHADORA3NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4313950-A Antireproductive tricyclic ortho-fused nitrogen containing compounds GRUPPO LEPETIT S.P.A. (IT) 1982-02-02 US disclosed
US-4275066-A 1,2,4-TRIAZOLO(5.1A)ISOINDOZE, TRIAZOLO(5.1A) ISOQUINOLINE OR 1,2,4,-TRIAZOLO (5.1A)(2) BENZAZEPINE CONTRACEPTIVES GRUPPO LEPETIT S.P.A. (IT) 1981-06-23 US disclosed