SCHEMBL11246376

SCHEMBL11246376

COC(=O)COc1ccc(CC[C@H](C)NCC(O)c2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 11/20 0.62
ADRB2 P07550 7/20 0.62
ADRB1 P08588 6/20 0.62
GLA P06280 1/20 0.62
ALDH1A1 P00352 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
KDM4E B2RXH2 3/20 0.53
GAA P10253 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
ADRA1A P35348 4/20 0.53
CYP2D6 P10635 3/20 0.53
ADRA1D P25100 3/20 0.53
ADRA1B P35368 3/20 0.53
CYP1A2 P05177 2/20 0.53
CYP2C19 P33261 2/20 0.53
CYP2C9 P11712 1/20 0.53
HTR1A P08908 2/20 0.50
ADRA2A P08913 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11251142 0.89 ADRB3 (0.77) ADRB3ADRB2ADRB1GLAADRA1A
SCHEMBL11247530 0.89 ADRB3 (0.77) ADRB3ADRB2ADRB1GLAADRA1A
SCHEMBL10562541 0.84 BCHE (0.69) ADRB3ADRB2ADRB1ALDH1A1MEN1
SCHEMBL10562535 0.84 BCHE (0.69) ADRB3ADRB2ADRB1ALDH1A1MEN1
Hydrochloric Acid SCHEMBL11477403 0.83 BCHE (0.67) ADRB3ADRB2ADRB1ALDH1A1MEN1
SCHEMBL10562146 0.83 ADRB2 (0.57) ADRB3ADRB2ADRB1ALDH1A1MEN1
Hydrochloric Acid SCHEMBL10564630 0.83 BCHE (0.67) ADRB3ADRB2ADRB1ALDH1A1MEN1
SCHEMBL10562158 0.83 ADRB2 (0.57) ADRB3ADRB2ADRB1ALDH1A1MEN1
Hydrochloric Acid SCHEMBL11477401 0.83 BCHE (0.67) ADRB3ADRB2ADRB1ALDH1A1MEN1
Ractopamine SCHEMBL352564 0.83 ADRB2 (0.68) ADRB3ADRB2ADRB1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US claimed
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US disclosed
EP-0023385-A1 Ethanamine derivatives, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-02-04 EP disclosed