SCHEMBL11246435

SCHEMBL11246435

CC(C)NC1CCc2c[nH]c3cccc(c23)C1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.49
OPRM1 P35372 2/20 0.47
MEN1 O00255 3/20 0.39
MAPT P10636 3/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP2D6 P10635 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
KDM4E B2RXH2 2/20 0.37
CYP3A4 P08684 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CYP1A2 P05177 1/20 0.37
THRB P10828 1/20 0.37
ALOX15 P16050 1/20 0.37
APEX1 P27695 1/20 0.37
MAPK1 P28482 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11206777 0.87 ADRB2 (0.45) ADRB2OPRM1MEN1MAPTKMT2A
SCHEMBL11239304 0.86 MEN1 (0.41) MEN1MAPTKMT2AALDH1A1CYP2D6
SCHEMBL11006874 0.86 MEN1 (0.41) MEN1MAPTKMT2AALDH1A1CYP2D6
SCHEMBL11240757 0.86 MEN1 (0.41) MEN1MAPTKMT2AALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL11246213 0.85 MEN1 (0.40) OPRM1MEN1MAPTKMT2AALDH1A1
SCHEMBL20131098 0.77 ADRB2 (0.56) ADRB2OPRM1CYP2D6
SCHEMBL11272560 0.76 ALDH1A1 (0.42) MEN1MAPTKMT2AALDH1A1CYP2D6
SCHEMBL11236653 0.76 CYP2D6 (0.39) MEN1MAPTKMT2AALDH1A1CYP2D6
SCHEMBL11260060 0.76 HTR2A (0.42) MEN1MAPTKMT2AALDH1A1CYP2D6
SCHEMBL10814023 0.75 MEN1 (0.46) MEN1MAPTKMT2AALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4335135-A 5 Amino-3,4,5,6 tetrahydro-1H-[-6-]cyclohept[c,d]indolols and a method for their use as hypotensives ROUSSEL UCLAF (FR) 1982-06-15 US disclosed