SCHEMBL11246471

SCHEMBL11246471

Cc1cc(-c2cnc(Cl)c(Br)c2)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 2/20 0.46
DYRK1A Q13627 3/20 0.44
AAK1 Q2M2I8 2/20 0.41
ALDH1A1 P00352 1/20 0.41
TLR8 Q9NR97 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
UHRF1 Q96T88 1/20 0.38
MAP4K4 O95819 1/20 0.38
HTT P42858 1/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
PIK3CD O00329 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11237788 0.83 AAK1 (0.49) PIK3CBDYRK1AAAK1TLR8TLR7
SCHEMBL7282401 0.79 PIK3CD (0.50) PIK3CBALDH1A1PIK3CDPIK3CAPIK3CG
SCHEMBL7272389 0.76 ALDH1A1 (0.60) PIK3CBDYRK1AAAK1ALDH1A1CYP3A4
SCHEMBL14934011 0.76 AAK1 (0.49) PIK3CBDYRK1AAAK1TLR8TLR7
SCHEMBL30308690 0.75 DYRK1A (0.65) PIK3CBDYRK1ACYP3A4CYP2D6PSEN1
SCHEMBL1896511 0.75 DYRK1A (0.65) PIK3CBDYRK1ACYP3A4CYP2D6PSEN1
SCHEMBL11377602 0.75 PIK3CB (0.58) PIK3CBPSEN1PSEN2APH1BNCSTN
SCHEMBL11153504 0.74 PIK3CB (0.72) PIK3CBAAK1PSEN1PSEN2APH1B
SCHEMBL11170792 0.74 TLR8 (0.60) PIK3CBDYRK1AAAK1TLR8TLR7
Iodide SCHEMBL9618570 0.73 DYRK1A (0.63) PIK3CBDYRK1ACYP3A4CYP2D6PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4351941-A Pyridinyl-pyridines STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4331672-A 5-(Pyridinyl)pyridine-2-hydrazines, their preparation and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed