SCHEMBL11248087

SCHEMBL11248087

CN(C)C(=O)Cc1ccc2c(c1)sc1ccc(Cl)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
MAPT P10636 1/20 0.40
KDM4E B2RXH2 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
F10 P00742 1/20 0.38
MAPK1 P28482 1/20 0.38
BCKDK O14874 1/20 0.38
MCL1 Q07820 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
SLC22A12 Q96S37 1/20 0.37
ALOX5 P09917 2/20 0.36
PIM1 P11309 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
ERCC1 P07992 1/20 0.35
ERCC4 Q92889 1/20 0.35
TSPO P30536 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11240017 0.83 KEAP1 (0.51) MAPTKDM4EKEAP1NFE2L2BCKDK
SCHEMBL11253511 0.83 KDM4E (0.42) MAPTKDM4EKEAP1NFE2L2F10
SCHEMBL11232073 0.82 SIRT1 (0.44) MAPTKDM4EKEAP1NFE2L2BCKDK
Methane SCHEMBL11235653 0.82 KEAP1 (0.50) MAPTKDM4EKEAP1NFE2L2BCKDK
SCHEMBL11237145 0.82 NPC1 (0.47) MAPTALDH1A1RAB9A
Butane SCHEMBL11246725 0.82 KEAP1 (0.47) MAPTKDM4EKEAP1NFE2L2MAPK1
Methane SCHEMBL11235493 0.81 SIRT1 (0.43) MAPTKDM4EKEAP1NFE2L2BCKDK
Methane SCHEMBL11228447 0.81 NPC1 (0.46) MAPTALDH1A1RAB9A
Butane SCHEMBL11229487 0.80 NPC1 (0.46) MAPTRAB9A
SCHEMBL11241148 0.80 KLK7 (0.36) MAPTKDM4EF10MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed