SCHEMBL11248154

SCHEMBL11248154

COc1ccc2c(c1)C(=O)C1(CCN(C)CC1)c1cc(Cl)ccc1O2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.42
SLC6A4 P31645 3/20 0.42
SLC6A3 Q01959 3/20 0.42
PPIB P23284 1/20 0.41
DRD2 P14416 6/20 0.40
DRD4 P21917 5/20 0.40
HRH1 P35367 3/20 0.40
HTR2A P28223 3/20 0.40
BACE1 P56817 5/20 0.40
CTSD P07339 3/20 0.40
HTR2C P28335 3/20 0.40
DRD1 P21728 2/20 0.38
DRD5 P21918 2/20 0.38
DRD3 P35462 2/20 0.38
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11243297 0.92 PPIB (0.45) PPIBDRD2DRD4HTR2ABACE1
SCHEMBL11246209 0.83 HRH1 (0.40) SLC6A2SLC6A4SLC6A3DRD2DRD4
SCHEMBL11248897 0.82 HRH1 (0.56) SLC6A2SLC6A4SLC6A3DRD2DRD4
Bromide SCHEMBL11473841 0.81 HRH1 (0.56) SLC6A2SLC6A4SLC6A3DRD2DRD4
SCHEMBL11245536 0.81 HRH1 (0.42) SLC6A2SLC6A4SLC6A3DRD2DRD4
SCHEMBL11435472 0.80 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3DRD2DRD4
SCHEMBL7681805 0.79 HRH4 (0.45) SLC6A2SLC6A4SLC6A3DRD2DRD4
Hydrochloric Acid SCHEMBL11400430 0.78 HRH4 (0.44) SLC6A2SLC6A4SLC6A3DRD2DRD4
SCHEMBL11257464 0.77 MAPK14 (0.41) PPIBDRD2DRD4BACE1CTSD
SCHEMBL11242210 0.77 HRH1 (0.41) SLC6A2SLC6A4SLC6A3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0016261-B1 SPIRO(DIBENZ(B,F)OXEPIN-PIPERIDINES) AND METHODS OF PREPARING SAME HOECHST AKTIENGESELLSCHAFT (DE) 1982-12-29 EP disclosed
US-4198418-A ANALGESICS, TRANQUILIZERS, ANTICONVULSANTS AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed