SCHEMBL11248247

SCHEMBL11248247

OCc1c(-c2ccccc2)nn(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
KDM4E B2RXH2 2/20 0.49
USP2 O75604 2/20 0.49
MAPT P10636 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
HSD17B10 Q99714 2/20 0.49
GMNN O75496 1/20 0.49
LMNA P02545 1/20 0.49
ESR1 P03372 1/20 0.49
TP53 P04637 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
ALOX12 P18054 1/20 0.49
NFKB1 P19838 1/20 0.49
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifezolac SCHEMBL11182574 0.83 KDM4E (0.51) KMT2ACYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL11724930 0.82 SMN1; SMN2 (0.54) KMT2AKDM4EUSP2MAPTNPSR1
SCHEMBL11731343 0.82 SMN1; SMN2 (0.49) KMT2AKDM4EUSP2MAPTNPSR1
SCHEMBL14747800 0.81 PTGS2 (0.50) CYP1A2CYP2C9CYP2C19SMN1; SMN2PTGS2
SCHEMBL11249543 0.80 CYP2C9 (0.47) KMT2ACYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL8122183 0.80 CYP2C9 (0.47) KMT2ACYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL11258179 0.80 CA1 (0.43) KMT2ACYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL27574894 0.78 CYP2C9 (0.58) KMT2ACYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL11258090 0.78 CYP2C9 (0.48) KMT2ACYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL11245216 0.78 KMT2A (0.48) KMT2ACYP1A2CYP2C9CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4325962-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIDYRETICS BYK-GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1982-04-20 US disclosed
US-4146721-A ANALGESICS, ANTIINFLAMMATORY AGENTS AND ANTIPYRETICS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1979-03-27 US disclosed