SCHEMBL14747800

SCHEMBL14747800

OCc1c(C(F)(F)F)nn(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.50
CACNA1G O43497 2/20 0.49
CACNA1H O95180 2/20 0.49
CACNA1I Q9P0X4 2/20 0.49
PTGS1 P23219 4/20 0.48
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14747606 0.91 PTGS2 (0.51) PTGS2CACNA1GCACNA1HCACNA1IPTGS1
SCHEMBL6351481 0.85 PTGS2 (0.73) PTGS2PTGS1
SCHEMBL3379848 0.82 CACNA1G (0.39) PTGS2CACNA1GCACNA1HCACNA1IPTGS1
SCHEMBL11248247 0.81 KMT2A (0.49) PTGS2CACNA1GCACNA1HCACNA1IPTGS1
SCHEMBL3383520 0.81 BRAF (0.43) PTGS2PTGS1SMN1; SMN2
SCHEMBL14747809 0.78 PTGS2 (0.71) PTGS2PTGS1CYP1A2CYP2C9CYP2C19
SCHEMBL8689175 0.78 F10 (0.49) PTGS2PTGS1
SCHEMBL14747815 0.77 PTGS2 (0.54) PTGS2PTGS1CYP1A2CYP2C9CYP2C19
SCHEMBL538098 0.75 CACNA1G (0.35) PTGS2CACNA1GCACNA1HCACNA1IPTGS1
SCHEMBL14747799 0.72 PTGS2 (0.47) PTGS2PTGS1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44048-E1 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-YL]benzenesulfonamide for the treatment of inflammation or an inflammation-associated disorder G.D. SEARLE LLC (US) 2013-03-05 US disclosed