SCHEMBL11248670

SCHEMBL11248670

O=C(O)c1ccc(NCc2cccc(Cl)c2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.58
RXRA P19793 2/20 0.57
RXRB P28702 2/20 0.57
RXRG P48443 2/20 0.57
MRGPRX4 Q96LA9 2/20 0.57
HDAC1 Q13547 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
HDAC3 O15379 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.51
ADRB2 P07550 1/20 0.51
ADRB1 P08588 1/20 0.51
ADRB3 P13945 1/20 0.51
POLB P06746 1/20 0.51
MAPT P10636 1/20 0.51
THRB P10828 1/20 0.51
TAS2R14 Q9NYV8 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
PTGER4 P35408 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4745951 0.88 FFAR1 (0.60) RXRARXRBRXRGADRB3
SCHEMBL13802457 0.87 MRGPRX4 (0.63) HIF1AMRGPRX4HDAC6HDAC8
SCHEMBL6840198 0.85 PPARA (0.60) RXRARXRBRXRGMRGPRX4POLB
SCHEMBL29080372 0.84 PTK2 (0.59) HIF1AHDAC1HDAC6HDAC3HDAC2
SCHEMBL30519428 0.84 PTK2 (0.59) HIF1AHDAC1HDAC6HDAC3HDAC2
SCHEMBL30687018 0.84 FFAR1 (0.65) ADRB2ADRB1ADRB3HDAC4MEF2D
SCHEMBL30687014 0.84 FFAR1 (0.65) ADRB2ADRB1ADRB3HDAC4MEF2D
SCHEMBL29129870 0.84 FFAR1 (0.65) ADRB2ADRB1ADRB3HDAC4MEF2D
SCHEMBL4748420 0.83 HIF1A (0.68) HIF1AMRGPRX4HDAC6HDAC8POLB
SCHEMBL27487037 0.83 HIF1A (0.69) HIF1AMRGPRX4HDAC6HDAC8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090155903-A1 PHARMACEUTICAL COMPOSITION AND METHOD MYRIAD GENETICS, INCORPORATED (US) 2009-06-18 US disclosed
US-20090155903-A1 PHARMACEUTICAL COMPOSITION AND METHOD MYRIAD GENETICS, INCORPORATED (US) 2009-06-18 US disclosed
US-4362892-A ARALKYLANILINES, ANTICHOLESTEROL AGENTS BEECHAM GROUP LIMITED (GB) 1982-12-07 US disclosed
US-4207330-A Method for treating hyperglycemia in mammals using arylamino benzoic acids THE DOW CHEMICAL COMPANY (US) 1980-06-10 US disclosed
US-4206145-A ALKANOYL-SUBSTITUTED ARALKYLAMINES BEECHAM GROUP LIMITED (GB) 1980-06-03 US disclosed
US-4143151-A METHOD FOR TREATING HYPERGLYCEMIA IN MAMMALS USING ARYLAMINO BENZOIC ACIDS THE DOW CHEMICAL COMPANY (US) 1979-03-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090155903-A1 PHARMACEUTICAL COMPOSITION AND METHOD APP, PSEN2, PSEN1 HIF1A 2788/4885RXRA 3288/4885RXRB 3134/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.