SCHEMBL29080372

SCHEMBL29080372

CNC(=O)c1ccc(NCc2cccc(Cl)c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.59
HDAC1 Q13547 6/20 0.56
IDH1 O75874 1/20 0.53
HDAC6 Q9UBN7 2/20 0.52
HDAC3 O15379 2/20 0.52
HDAC2 Q92769 2/20 0.52
HDAC8 Q9BY41 1/20 0.48
SCD O00767 1/20 0.47
NCOR2 Q9Y618 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
HDAC4 P56524 1/20 0.46
MEF2D Q14814 1/20 0.46
NPC1 O15118 1/20 0.46
GPR17 Q13304 1/20 0.46
HIF1A Q16665 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30519428 1.00 PTK2 (0.59) PTK2HDAC1IDH1HDAC6HDAC3
SCHEMBL11248670 0.84 HIF1A (0.58) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL11253249 0.80 TRPV1 (0.64) CA1CA2NPC1HIF1A
SCHEMBL11510712 0.78 HDAC4 (0.54) HDAC1HDAC6HDAC3HDAC2HDAC4
SCHEMBL8234606 0.77 HTT (0.62) NPC1
SCHEMBL30687018 0.77 FFAR1 (0.65) HDAC4MEF2D
SCHEMBL30687014 0.77 FFAR1 (0.65) HDAC4MEF2D
SCHEMBL29129870 0.77 FFAR1 (0.65) HDAC4MEF2D
SCHEMBL30687017 0.76 FFAR1 (0.50) HDAC1HDAC6HDAC3HDAC2HDAC4
SCHEMBL3241843 0.76 NPC1 (0.63) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116554153-A Tertiary amide compounds and medical use thereof 中国人民解放军军事科学院军事医学研究院 2023-08-08 CN disclosed