SCHEMBL11249334

SCHEMBL11249334

CN(C)c1ccccc1-c1nccc2c(CC(=O)O)cccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.44
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
CNR2 P34972 1/20 0.38
CYP1A2 P05177 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
PPARG P37231 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
PTGDR2 Q9Y5Y4 4/20 0.36
AKR1B1 P15121 1/20 0.36
PTGER1 P34995 1/20 0.34
PTGER4 P35408 1/20 0.34
PTGER3 P43115 1/20 0.34
PTGER2 P43116 1/20 0.34
EDNRA P25101 1/20 0.33
SLC40A1 Q9NP59 1/20 0.33
AR P10275 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11252493 0.84 TDP1 (0.48) TDP1RXRARXRBCYP1A2KDM4E
SCHEMBL11258381 0.81 TDP1 (0.48) TDP1CYP1A2KDM4EMAPTPTGDR2
SCHEMBL11257137 0.81 TDP1 (0.48) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11261730 0.81 TDP1 (0.44) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11262924 0.80 HPGD (0.36) CNR2CYP1A2KDM4EMAPTEDNRA
SCHEMBL11250186 0.79 PTGDR2 (0.43) TDP1RXRARXRBCNR2CYP1A2
SCHEMBL11251835 0.79 TDP1 (0.54) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL31644190 0.78 TDP1 (0.56) TDP1RXRARXRBCYP1A2MAPT
SCHEMBL11257961 0.77 KDM4E (0.42) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11262890 0.77 CNR2 (0.38) TDP1CNR2KDM4EMAPTSLC40A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed