SCHEMBL11261730

SCHEMBL11261730

CNc1ccccc1-c1nccc2c(CC(=O)O)cccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.44
PPARG P37231 2/20 0.43
NR1H2 P55055 2/20 0.43
NR1H3 Q13133 2/20 0.43
PARP14 Q460N5 1/20 0.41
PTGS2 P35354 4/20 0.41
CXCL8 P10145 3/20 0.40
ACHE P22303 1/20 0.40
TTR P02766 2/20 0.39
NR1H4 Q96RI1 2/20 0.39
AKR1B10 O60218 1/20 0.39
UGT1A9 O60656 1/20 0.39
TRPA1 O75762 1/20 0.39
ABCB11 O95342 1/20 0.39
MT-CO2 P00403 1/20 0.39
ALB P02768 1/20 0.39
UGT1A6 P19224 1/20 0.39
UGT1A1 P22309 1/20 0.39
PTGS1 P23219 1/20 0.39
CXCR1 P25024 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11252493 0.84 TDP1 (0.48) TDP1PPARGNR1H2NR1H3PTGS2
SCHEMBL11258381 0.81 TDP1 (0.48) TDP1PTGS2CXCL8TTRNR1H4
SCHEMBL11257137 0.81 TDP1 (0.48) TDP1PPARGNR1H2NR1H3CXCL8
SCHEMBL11249334 0.81 TDP1 (0.44) TDP1PPARGNR1H2NR1H3PTGS2
SCHEMBL11259158 0.79 TDP1 (0.42) TDP1PPARGNR1H2NR1H3KDM4E
SCHEMBL11251835 0.79 TDP1 (0.54) TDP1PPARGNR1H2NR1H3KDM4E
SCHEMBL11285948 0.77 NR1H2 (0.42) TDP1PPARGNR1H2NR1H3KDM4E
SCHEMBL11266224 0.77 CXCL8 (0.41) TDP1PARP14PTGS2CXCL8ACHE
SCHEMBL11246786 0.74 LMNA (0.48) TDP1PPARGNR1H2NR1H3KDM4E
SCHEMBL11311256 0.73 TDP1 (0.53) TDP1PPARGNR1H2NR1H3PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed