SCHEMBL11250945

SCHEMBL11250945

Cc1cc(Br)ccc1NC(=N)NC(N)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.51
MAPT P10636 6/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
DHODH Q02127 1/20 0.47
NPY1R P25929 1/20 0.46
NPY2R P49146 1/20 0.46
ALDH1A1 P00352 4/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
POLB P06746 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11259170 0.88 POLB (0.43) SIGMAR1MAPTMEN1KMT2ADHODH
SCHEMBL11405358 0.88 SIGMAR1 (0.54) SIGMAR1MAPTMEN1KMT2ADHODH
SCHEMBL11578514 0.84 NPC1 (0.43) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL11579511 0.84 MEN1 (0.56) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL18324579 0.84 SIGMAR1 (0.59) SIGMAR1MAPTMEN1KMT2ADHODH
SCHEMBL11252261 0.84 MAPK1 (0.48) MAPTMEN1KMT2ANPY1RNPY2R
SCHEMBL6719185 0.84 SIGMAR1 (0.56) SIGMAR1MAPTMEN1KMT2ADHODH
SCHEMBL11581488 0.82 MAPT (0.38) MAPTALDH1A1NPC1RAB9AHPGD
SCHEMBL11266958 0.82 MAPK1 (0.51) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL11254202 0.82 ALDH1A1 (0.46) SIGMAR1MAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4115564-A Treatment of diarrhea with amidinoureas WILLIAM H. RORER, INC. (US) 1978-09-19 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed