SCHEMBL11253003

SCHEMBL11253003

O=C(O)c1ccc2c(c1)sc1cc(Cl)ccc12.[KH]

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCKDK O14874 2/20 0.58
MCL1 Q07820 1/20 0.58
RXFP1 Q9HBX9 1/20 0.58
TTR P02766 4/20 0.50
TSHR P16473 2/20 0.48
ALOX15 P16050 1/20 0.48
SRD5A2 P31213 4/20 0.46
SRD5A1 P18405 1/20 0.46
TBXAS1 P24557 1/20 0.44
MAP2K4 P45985 1/20 0.43
PRSS12 P56730 1/20 0.43
SPR P35270 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30414903 0.87 KDM4E (0.48) BCKDKMCL1RXFP1TSHRSRD5A2
SCHEMBL204515 0.87 KDM4E (0.48) BCKDKMCL1RXFP1TSHRSRD5A2
SCHEMBL11247121 0.84 BCKDK (0.51) BCKDKMCL1RXFP1TTRTSHR
SCHEMBL30414825 0.83 KDM4E (0.46) BCKDKMCL1RXFP1TSHRSRD5A2
SCHEMBL14020124 0.83 KDM4E (0.60) BCKDKMCL1RXFP1TTRTSHR
Potassium Ion SCHEMBL11253001 0.81 CA1 (0.50) BCKDKMCL1RXFP1TTRPRSS12
SCHEMBL11244432 0.81 CYP1A2 (0.53) MCL1TTRTSHRALOX15NPC1
SCHEMBL4922527 0.79 BCKDK (0.53) BCKDKMCL1RXFP1MEN1KMT2A
SCHEMBL31228783 0.79 BCKDK (0.53) BCKDKMCL1RXFP1MEN1KMT2A
SCHEMBL29762008 0.79 CYP1A2 (0.54) MCL1TTRTSHRALOX15NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed