SCHEMBL1125436

SCHEMBL1125436

Nc1cccc(-c2c(Cc3ccccc3)c(C(F)(F)F)nc3ccccc23)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.39
BACE1 P56817 1/20 0.38
CCNE2 O96020 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
ADORA2A P29274 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ENPP1 P22413 2/20 0.37
ELANE P08246 1/20 0.37
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
CYP17A1 P05093 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
MAOA P21397 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29834189 0.74 ESR1 (0.56) ADORA2ANPC1RAB9AMAOAESR1
SCHEMBL601251 0.74 ESR1 (0.56) ADORA2ANPC1RAB9AMAOAESR1
SCHEMBL16633300 0.72 MAOA (0.46) APPCCNE2CCNE1CDK2ENPP1
SCHEMBL1124687 0.69 NR1H2 (0.68)
SCHEMBL29253732 0.67 CYP1A2 (0.53) APPADORA2ACYP3A4CYP1A2CYP2D6
SCHEMBL27651468 0.65 ESR1 (0.51) NPC1RAB9AMAOAESR1KDM4E
SCHEMBL31326856 0.65 TLR7 (0.50) APPBACE1CCNE2CCNE1CDK2
SCHEMBL28027243 0.65 ENPP1 (0.48) ENPP1ESR1KDM4EMAPTSMN1; SMN2
SCHEMBL31326858 0.65 TLR7 (0.50) APPBACE1CCNE2CCNE1CDK2
SCHEMBL12337344 0.64 MAOA (0.64) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2284157-A1 Quinolines useful in treating cardiovascular disease Wyeth (US) 2011-02-16 EP disclosed