SCHEMBL11255856

SCHEMBL11255856

Clc1cccc2c(-c3ccccc3)nccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.48
CYP2A6 P11509 3/20 0.48
TDO2 P48775 3/20 0.47
HTR2B P41595 1/20 0.47
HTR5A P47898 1/20 0.47
L3MBTL1 Q9Y468 3/20 0.43
NPSR1 Q6W5P4 3/20 0.43
ALDH1A1 P00352 2/20 0.43
IDO1 P14902 2/20 0.43
ADORA2A P29274 1/20 0.43
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
NQO2 P16083 1/20 0.42
NR4A2 P43354 2/20 0.41
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
GPR55 Q9Y2T6 1/20 0.40
DHODH Q02127 1/20 0.39
GLA P06280 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11265968 0.84 ALDH1A1 (0.44) CYP1A2CYP2A6TDO2L3MBTL1NPSR1
SCHEMBL30631719 0.81 PLG (0.54) TDO2HTR2BHTR5AL3MBTL1NPSR1
SCHEMBL23095358 0.79 ALDH1A1 (0.48) CYP1A2CYP2A6L3MBTL1NPSR1ALDH1A1
SCHEMBL26185762 0.78 TDO2 (0.42) TDO2HTR2BHTR5AL3MBTL1NPSR1
SCHEMBL11976465 0.78 NQO2 (0.49) CYP1A2CYP2A6TDO2HTR2BHTR5A
SCHEMBL13169304 0.78 PLG (0.51) TDO2HTR2BHTR5AL3MBTL1NPSR1
SCHEMBL3146190 0.78 TDO2 (0.47) CYP1A2TDO2HTR2BHTR5AL3MBTL1
SCHEMBL15712262 0.78 ALDH1A1 (0.48) TDO2HTR2BHTR5AL3MBTL1NPSR1
SCHEMBL11259942 0.77 TDO2 (0.44) TDO2HTR2BHTR5AL3MBTL1NPSR1
SCHEMBL11100168 0.77 PDE3B (0.53) CYP1A2TDO2HTR2BHTR5AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed