SCHEMBL11258499

SCHEMBL11258499

CNC(C)CC(c1ccccc1)c1ccc(Br)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.52
SLC6A3 Q01959 3/20 0.51
CHRM2 P08172 3/20 0.51
CHRM1 P11229 2/20 0.51
HRH1 P35367 2/20 0.51
ADRA1A P35348 2/20 0.51
CACNA1F O60840 1/20 0.51
ADRA2B P18089 1/20 0.51
CHRM3 P20309 1/20 0.51
OPRK1 P41145 1/20 0.51
CACNA1D Q01668 1/20 0.51
KCNH2 Q12809 1/20 0.51
CACNA1S Q13698 1/20 0.51
CACNA1C Q13936 1/20 0.51
SCN5A Q14524 1/20 0.51
SLC6A4 P31645 3/20 0.47
SLC6A2 P23975 2/20 0.47
TAAR1 Q96RJ0 3/20 0.44
SIGMAR1 Q99720 2/20 0.44
SLC18A2 Q05940 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281996 0.89 HRH1 (0.62) HTR2ASLC6A3CHRM2CHRM1HRH1
Hydrochloric Acid SCHEMBL7274257 0.87 HRH1 (0.60) HTR2ASLC6A3CHRM2CHRM1HRH1
SCHEMBL11249446 0.78 HTR2A (0.60) HTR2ASLC6A3CHRM2CHRM1HRH1
SCHEMBL1979887 0.76 SLC6A4 (0.65) HTR2ASLC6A3CHRM2CHRM1HRH1
SCHEMBL11241825 0.74 SMN1; SMN2 (0.45) CNR1SMN1; SMN2ALDH1A1LMNACYP3A4
SCHEMBL17802362 0.72 HTR2A (0.63) HTR2ASLC6A3CHRM2CHRM1HRH1
SCHEMBL16260323 0.72 HTR2A (0.56) HTR2ASLC6A3CHRM2CHRM1SLC6A4
SCHEMBL17685575 0.72 TAAR1 (0.48) HTR2ASLC6A3CHRM2CHRM1HRH1
SCHEMBL1291652 0.72 LMNA (0.52) HTR2ASLC6A3CHRM2CHRM1HRH1
SCHEMBL5468813 0.70 LMNA (0.61) HTR2ASLC6A3CHRM2CHRM1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000322-B1 COMPOUNDS HAVING AN ANTI-DEPRESSIVE OR TRANQUILIZING ACTIVITY, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION Astra Läkemedel Aktiebolag (SE) 1982-05-05 EP disclosed
EP-0028682-A2 Intermediates useful at the preparation of compounds having anti-depressive or tranquilizing activity Astra Läkemedel Aktiebolag (SE) 1981-05-20 EP disclosed