SCHEMBL7281996

SCHEMBL7281996

CNC(C)CC(c1ccccc1)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.62
ADRA1A P35348 4/20 0.62
CHRM2 P08172 3/20 0.62
SLC6A3 Q01959 3/20 0.62
KCNH2 Q12809 3/20 0.62
CHRM1 P11229 2/20 0.62
ADRA2B P18089 2/20 0.62
OPRK1 P41145 2/20 0.62
CACNA1C Q13936 2/20 0.62
SCN5A Q14524 2/20 0.62
CACNA1F O60840 1/20 0.62
CHRM3 P20309 1/20 0.62
CACNA1D Q01668 1/20 0.62
CACNA1S Q13698 1/20 0.62
TAAR1 Q96RJ0 5/20 0.54
SIGMAR1 Q99720 2/20 0.54
SLC18A2 Q05940 1/20 0.54
HTR2A P28223 5/20 0.48
CYP3A4 P08684 3/20 0.47
CYP2D6 P10635 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7274257 0.98 HRH1 (0.60) HRH1ADRA1ACHRM2SLC6A3KCNH2
SCHEMBL11258499 0.89 HTR2A (0.52) HRH1ADRA1ACHRM2SLC6A3KCNH2
SCHEMBL17685575 0.81 TAAR1 (0.48) HRH1ADRA1ACHRM2SLC6A3KCNH2
SCHEMBL1291652 0.81 LMNA (0.52) HRH1ADRA1ACHRM2SLC6A3KCNH2
SCHEMBL14415598 0.79 CACNA1F (0.42) HRH1ADRA1ACHRM2SLC6A3KCNH2
Terodiline SCHEMBL9008621 0.77 HRH1 (1.00) HRH1ADRA1ACHRM2SLC6A3KCNH2
Terodiline SCHEMBL78908 0.77 HRH1 (1.00) HRH1ADRA1ACHRM2SLC6A3KCNH2
SCHEMBL9493121 0.75 HRH1 (0.54) HRH1ADRA1ACHRM2SLC6A3KCNH2
Terodiline SCHEMBL121864 0.75 HRH1 (0.96) HRH1ADRA1ACHRM2SLC6A3KCNH2
SCHEMBL15130931 0.75 ADRA1A (0.55) HRH1ADRA1ACHRM2SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4968832-A INTERMEDIATES FOR CORONARY DILATORS RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1990-11-06 US disclosed
US-4772621-A Antihypertensive diphenylpropyl aminopropyl ester of 1,4-dihydro-2,6-dimethyl-pyridine-3,5-dicarboxylic acid RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1988-09-20 US disclosed
US-4705797-A HYPOTENSIVE AGENTS, VASODILATORS RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1987-11-10 US disclosed
EP-0153016-A2 Asymmetrical diesters of 1,4-dihydro-2,6-dimethyl-pyridine-3,5-dicarboxylic acid RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1985-08-28 EP disclosed
US-3946063-A 2,3,4,5,6-PENTAFLUOROBENZYL CHLOROFORMATE PIERCE CHEMICAL COMPANY (US) 1976-03-23 US disclosed