SCHEMBL11258960

SCHEMBL11258960

O=CC1C(=O)C=Cc2cc(Br)ccc21

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 1/20 0.32
EDNRB P24530 1/20 0.32
EDNRA P25101 1/20 0.32
ERN1 O75460 1/20 0.31
HSP90AA1 P07900 1/20 0.31
TLR9 Q9NR96 1/20 0.31
S100A4 P26447 1/20 0.31
CA12 O43570 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5823531 0.74 CYP2D6 (0.41) ALDH1A1
SCHEMBL998511 0.71 EDNRB (0.44) CYP1A2MAPK1EDNRBEDNRAHSP90AA1
SCHEMBL28092444 0.70 CYP1A2 (0.43) CYP1A2MAPK1ALDH1A1EDNRBEDNRA
SCHEMBL27808522 0.68 ALDH1A1 (0.32) ALDH1A1ERN1
SCHEMBL18748412 0.66 S100A4 (0.41) CYP1A2MAPK1ALDH1A1EDNRBEDNRA
SCHEMBL28507942 0.66 BRD4 (0.32) ALDH1A1
SCHEMBL28880613 0.64 S100A4 (0.41) CYP1A2MAPK1ALDH1A1EDNRBEDNRA
SCHEMBL27716951 0.63 CYP1A2 (0.53) CYP1A2MAPK1ALDH1A1EDNRBEDNRA
SCHEMBL29954649 0.62 TP53 (0.46) ALDH1A1CA12CA2CA9
SCHEMBL28237453 0.62 KDM1A (0.32) CYP1A2MAPK1EDNRBEDNRAHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0010740-B1 SPIRODIPYRANES AND THEIR USE AS COLOUR FORMERS IN COPYING PROCESSES BASF Aktiengesellschaft (DE) 1982-04-21 EP disclosed
EP-0010740-A1 Spirodipyranes and their use as colour formers in copying processes BASF Aktiengesellschaft (DE) 1980-05-14 EP disclosed