SCHEMBL11260412

SCHEMBL11260412

CC(COc1ccccc1)NCC(O)COc1cccc2[nH]ncc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.51
ADRB1 P08588 7/20 0.51
ADRB3 P13945 6/20 0.51
CYP2D6 P10635 5/20 0.51
HTR1A P08908 7/20 0.50
CYP1A2 P05177 5/20 0.50
ALDH1A1 P00352 5/20 0.50
LMNA P02545 4/20 0.50
HTR2C P28335 4/20 0.50
DRD3 P35462 4/20 0.50
TSHR P16473 3/20 0.50
MAPK1 P28482 3/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 2/20 0.50
TP53 P04637 2/20 0.50
NFKB1 P19838 2/20 0.50
HTR1B P28222 2/20 0.50
ADRA1A P35348 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11267040 0.82 DRD2 (0.59) ADRB2ADRB1ADRB3CYP2D6HTR1A
SCHEMBL11155478 0.76 NR2E1 (0.58) ADRB2ADRB1ADRB3CYP2D6HTR1A
SCHEMBL11270229 0.76 ADRB2 (0.43) ADRB2ADRB1ADRB3CYP2D6HTR1A
SCHEMBL11270462 0.76 ADRB2 (0.48) ADRB2ADRB1ADRB3CYP2D6HTR1A
Hydrochloric Acid SCHEMBL10605116 0.75 ADRB2 (0.54) ADRB2ADRB1ADRB3CYP2D6HTR1A
SCHEMBL11146826 0.75 DRD2 (0.55) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL11266544 0.74 ADRB2 (0.67) ADRB2ADRB1ADRB3HTR1ALMNA
SCHEMBL17738298 0.74 DRD4 (0.51) ADRB2ADRB1ADRB3CYP2D6HTR1A
SCHEMBL10934121 0.74 MEN1 (0.48) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL11226058 0.73 SLC6A2 (0.71) ADRB2ADRB1ADRB3CYP2D6HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4346093-A CARDIOVASCULAR DISORDERS BOEHRINGER MANNHEIM GMBH (DE) 1982-08-24 US disclosed