SCHEMBL11260792

SCHEMBL11260792

CCCC(C)c1nccc2c(CC(=O)O)cccc12

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
CYP1A2 P05177 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
PPARG P37231 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
AKR1B1 P15121 1/20 0.34
GLA P06280 1/20 0.33
STING1 Q86WV6 1/20 0.33
ABCB1 P08183 1/20 0.33
CDC25A P30304 1/20 0.33
CMA1 P23946 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
POLB P06746 2/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11249938 0.90 TDP1 (0.45) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11261355 0.86 TDP1 (0.50) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11250215 0.83 TDP1 (0.46) TDP1CYP1A2KDM4EMAPTPPARG
Formamide SCHEMBL11440222 0.81 TDP1 (0.44) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11249116 0.76 TDP1 (0.47) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11263624 0.75 TDP1 (0.44) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11248912 0.75 TDP1 (0.50) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11311256 0.75 TDP1 (0.53) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11251937 0.75 TDP1 (0.46) TDP1CYP1A2KDM4EMAPTPPARG
SCHEMBL11261670 0.74 ALDH1A1 (0.45) TDP1CYP1A2KDM4EMAPTPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed