SCHEMBL11261355

SCHEMBL11261355

CC(C)c1nccc2c(CC(=O)O)cccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
CYP1A2 P05177 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
AKR1B1 P15121 1/20 0.40
NR1H2 P55055 2/20 0.39
NR1H3 Q13133 2/20 0.39
PPARG P37231 1/20 0.39
GLA P06280 1/20 0.37
STING1 Q86WV6 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
POLB P06746 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.36
PTGS2 P35354 1/20 0.36
DUSP3 P51452 1/20 0.36
PTPN5 P54829 1/20 0.36
PTPN11 Q06124 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formamide SCHEMBL11440222 0.93 TDP1 (0.44) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11249938 0.89 TDP1 (0.45) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11250215 0.87 TDP1 (0.46) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11260792 0.86 TDP1 (0.43) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11255746 0.84 ALDH1A1 (0.40) KDM4ESMN1; SMN2ALDH1A1
SCHEMBL14755876 0.82 KDM4E (0.59) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11257657 0.82 LMNA (0.46) KDM4EMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL11254420 0.82 PKM (0.45) TDP1KDM4EMAPTSMN1; SMN2ALDH1A1
SCHEMBL11311256 0.81 TDP1 (0.53) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11251937 0.81 TDP1 (0.46) TDP1CYP1A2KDM4EMAPTAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
US-4329288-A CONTRAGESTATIONAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1982-05-11 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed