SCHEMBL11261802

SCHEMBL11261802

CC(C)(Oc1ccc2c(-c3ccncc3)c3n(c2c1)CCCCC3)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 2/20 0.38
TP53 P04637 2/20 0.35
PPARG P37231 4/20 0.35
SLC22A12 Q96S37 1/20 0.35
PPARA Q07869 6/20 0.35
CYP2C19 P33261 3/20 0.35
MEN1 O00255 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP2C9 P11712 2/20 0.35
PTPN7 P35236 1/20 0.35
DUSP3 P51452 1/20 0.35
PTPN12 Q05209 1/20 0.35
PTPN22 Q9Y2R2 1/20 0.35
GAA P10253 2/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11260420 0.92 GAA (0.39) TBXAS1TP53PPARGSLC22A12PPARA
SCHEMBL11269886 0.91 GAA (0.38) TBXAS1TP53PPARGSLC22A12PPARA
SCHEMBL11269896 0.91 GAA (0.38) TBXAS1TP53PPARGSLC22A12PPARA
SCHEMBL11264489 0.88 GAA (0.42) TP53PPARGPPARACYP1A2CYP3A4
SCHEMBL11269891 0.82 HTR6 (0.38) TP53CYP2C19MEN1CYP1A2CYP3A4
SCHEMBL11255435 0.80 GAA (0.46) TP53PPARGPPARACYP1A2CYP3A4
SCHEMBL11267432 0.79 GAA (0.45) TP53PPARGPPARACYP1A2CYP3A4
SCHEMBL11271278 0.79 PPARA (0.36) PPARGPPARACYP2C19MEN1CYP1A2
SCHEMBL11262244 0.76 GAA (0.42) CYP2C19MEN1CYP1A2CYP3A4KMT2A
SCHEMBL11500212 0.72 GAA (0.47) CYP2C19MEN1CYP1A2CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0015523-B1 INDOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE FOR MEDICAMENTS Dr. Karl Thomae GmbH (DE) 1982-10-13 EP disclosed
US-4343811-A ATHEROSCLEROSIS BOEHRINGER INGELHEIM GMBH (DE) 1982-08-10 US disclosed
EP-0015523-A1 Indole derivatives, their preparation and their use for medicaments Dr. Karl Thomae GmbH (DE) 1980-09-17 EP disclosed