SCHEMBL11271278

SCHEMBL11271278

Cc1cc2c(c(C)c1OC(C)(C)C(=O)O)c(-c1ccncc1)c1n2CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 16/20 0.36
PPARG P37231 14/20 0.36
PPARD Q03181 12/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
MEN1 O00255 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11261642 0.89 ALDH1A1 (0.38) PPARACYP1A2CYP2C9MEN1CYP3A4
SCHEMBL11260420 0.79 GAA (0.39) PPARAPPARGPPARDCYP1A2CYP2C9
SCHEMBL11261802 0.79 TBXAS1 (0.38) PPARAPPARGPPARDCYP1A2CYP2C9
SCHEMBL11267995 0.79 ADORA3 (0.40) CYP1A2CYP2C9MEN1CYP3A4CYP2C19
SCHEMBL11269896 0.78 GAA (0.38) PPARAPPARGPPARDCYP1A2CYP2C9
SCHEMBL11269891 0.70 HTR6 (0.38) CYP1A2CYP2C9MEN1CYP3A4CYP2C19
SCHEMBL11264489 0.70 GAA (0.42) PPARAPPARGCYP1A2CYP3A4KMT2A
SCHEMBL11255435 0.70 GAA (0.46) PPARAPPARGCYP1A2CYP3A4
SCHEMBL11267432 0.69 GAA (0.45) PPARAPPARGCYP1A2CYP3A4
SCHEMBL11262244 0.64 GAA (0.42) CYP1A2CYP2C9MEN1CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0015523-B1 INDOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE FOR MEDICAMENTS Dr. Karl Thomae GmbH (DE) 1982-10-13 EP disclosed