SCHEMBL11265026

SCHEMBL11265026

CCOc1ccc(-c2nc[nH]c2-c2ccc(F)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.61
MAPK13 O15264 1/20 0.61
RAF1 P04049 1/20 0.61
MAPK9 P45984 1/20 0.61
MAPK12 P53778 1/20 0.61
MAPK11 Q15759 1/20 0.61
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53
BRD4 O60885 1/20 0.52
KDM4E B2RXH2 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
CACNA2D1 P54289 1/20 0.47
IDO1 P14902 1/20 0.44
TNIK Q9UKE5 1/20 0.44
NR3C2 P08235 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
MAPK10 P53779 1/20 0.43
SCN9A Q15858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10992179 0.84 MAPK14 (0.83) MAPK14MAPK13RAF1MAPK9MAPK12
Hydrochloric Acid SCHEMBL30023185 0.82 MAPK14 (0.80) MAPK14MAPK13RAF1MAPK9MAPK12
SCHEMBL7087770 0.77 MAPK14 (0.67) MAPK14MAPK13RAF1MAPK9MAPK12
SCHEMBL4434902 0.76 MAPK14 (1.00) MAPK14MAPK13RAF1MAPK9MAPK12
SCHEMBL6423292 0.76 MAPK14 (1.00) MAPK14MAPK13RAF1MAPK9MAPK12
SCHEMBL1173733 0.76 MAPT (0.58) MAPK14MAPK13RAF1MAPK9MAPK12
SCHEMBL1547683 0.75 NQO1 (0.74) KDM4EMAPTALDH1A1CYP1A2CYP2D6
SCHEMBL5698694 0.73 MAPK14 (0.61) MAPK14MAPK13RAF1MAPK9MAPK12
Ammonia Solution, Strong SCHEMBL322908 0.73 NQO1 (0.70) KDM4ECACNA2D1ALDH1A1CYP1A2CYP2D6
SCHEMBL11273419 0.72 LMNA (0.52) MAPK14MAPK13MAPK9MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0008755-B1 ANTIINFLAMMATORY 4,5-DIARYL-2-NITROIMIDAZOLES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-04-21 EP disclosed
US-4199592-A Antiinflammatory 4,5-diaryl-2-nitroimidazoles E. I. DU PONT DE NEMOURS AND COMPANY (US) 1980-04-22 US disclosed
EP-0008755-A1 Antiinflammatory 4,5-diaryl-2-nitroimidazoles, method for their preparation and pharmaceutical composition containing them E.I. DU PONT DE NEMOURS AND COMPANY (US) 1980-03-19 EP disclosed