SCHEMBL1173733

SCHEMBL1173733

COc1ccc(-c2nc[nH]c2-c2ccc(OC)cc2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.58
KDM4E B2RXH2 2/20 0.58
CYP3A4 P08684 1/20 0.58
ADORA3 P0DMS8 2/20 0.53
IDO1 P14902 4/20 0.52
MAPK13 O15264 1/20 0.51
RAF1 P04049 1/20 0.51
MAPK9 P45984 1/20 0.51
MAPK12 P53778 1/20 0.51
MAPK11 Q15759 1/20 0.51
MAPK14 Q16539 1/20 0.51
ADORA1 P30542 1/20 0.48
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NOX1 Q9Y5S8 1/20 0.46
HPGD P15428 1/20 0.45
CLK4 Q9HAZ1 1/20 0.44
CCNB2 O95067 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Imidazole SCHEMBL8030609 0.87 MAPK14 (0.48) MAPTKDM4ECYP3A4ADORA3IDO1
SCHEMBL9744537 0.83 IDO1 (0.43) MAPTKDM4ECYP3A4ADORA3IDO1
SCHEMBL10959629 0.80 PDE10A (0.59) MAPTKDM4ECYP3A4ADORA3IDO1
SCHEMBL24278328 0.79 MAPT (0.51) MAPTKDM4ECYP3A4ADORA3IDO1
SCHEMBL11834419 0.79 KDM4E (0.64) MAPTKDM4ECYP3A4ADORA3IDO1
SCHEMBL15664736 0.77 IDO1 (0.46) MAPTKDM4ECYP3A4IDO1MAPK13
SCHEMBL30014823 0.76 IDO1 (0.56) MAPTKDM4ECYP3A4IDO1MAPK13
SCHEMBL10355401 0.76 SMN1; SMN2 (0.40) MAPTKDM4EADORA3IDO1KMT2A
SCHEMBL11265026 0.76 MAPK14 (0.61) MAPTKDM4ECYP3A4IDO1MAPK13
SCHEMBL10989572 0.76 KDM4E (0.60) MAPTKDM4ECYP3A4IDO1MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117946203-A Glycyrrhetinic acid-gold complex and preparation method and application thereof 南京中医药大学 2024-04-30 CN claimed
CN-117946203-A Glycyrrhetinic acid-gold complex and preparation method and application thereof 南京中医药大学 2024-04-30 CN disclosed
CN-110551156-B Specific group-modified N1, N3-substituted 4,5-diaryl imidazole ring carbene rhodium complex and preparation method and application thereof 南京中医药大学 2022-11-25 CN disclosed
US-7888118-B2 induces differentiation of myoblasts or muscle fiber into neuron cells; drug screening; useful for treatment of neurodegenerative disorders, such as stroke, spinal cord injury, Parkinson's and Alzheimer's diseases; 2-{2-[5-(3-chlorophenyl)]furanyl}-4,5-bis(4-methoxyphenyl)imidazole (Neurodazine 1) INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY (KR) 2011-02-15 US disclosed
US-20100184097-A1 4,5-BIS(4-METHOXYPHENYL)IMIDAZOLE COMPOUND INDUCING DIFFERENTIATION OF MYOBLASTS OR MUSCLE FIBERS INTO NEURON CELLS, A PHARMACEUTICAL COMPOSITION INCLUDING SAID COMPOUND, A METHOD OF INDUCING NEURON CELLS DIFFERENTIATION AND A SCREENING METHOD FOR IDENTIFYING ADDITIONAL COMPOUND USEFUL FOR INDUCING NEURON CELLS DIFFERENTIATION INDUSTRY-ACADEMIC CORPORATION FOUNDATION, YONSEI UNIVERSITY (KR) 2010-07-22 US disclosed
US-7718685-B2 4,5-bis(4-methoxyphenyl)imidizole compound inducing differentiation of myoblasts or muscle fibers and pharmaceutical compositions including said compound INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY (KR) 2010-05-18 US disclosed
US-7718685-B2 4,5-bis(4-methoxyphenyl)imidizole compound inducing differentiation of myoblasts or muscle fibers and pharmaceutical compositions including said compound INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY (KR) 2010-05-18 US disclosed
US-20050276764-A1 Topical use of bis-arylimidazo[1,2-a]thiolane derivatives BEIERSDORF AG 2005-12-15 US disclosed
WO-2000019994-A9 ESTROGEN RECEPTOR LIGANDS UNIV ILLINOIS (US) 2000-08-31 WO disclosed
EP-0626969-B1 CoA-IT AND PAF INHIBITORS SMITHKLINE BEECHAM CORP (US) 2000-05-24 EP disclosed
US-4431722-A POLYCYCLIC QUINONE PIGMENT DISPERSED IN A RESIN BINDER AS CHARGE GENERATING LAYER; ANTIFOGGING AGENTS KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1984-02-14 US disclosed
US-4402960-A Antiinflammatory imidazole derivatives SCHERING AKTIENGESELLSCHAFT (DE) 1983-09-06 US disclosed
EP-0010361-B1 BIS-IMIDAZOLES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITHKLINE BECKMAN CORPORATION (US) 1983-04-27 EP disclosed
US-4372964-A ANAGESIC, ANTIARTHRITIC E. I. DU PONT DE NEMOURS AND COMPANY (US) 1983-02-08 US disclosed
EP-0011115-B1 ANTIINFLAMMATORY 2-SUBSTITUTED-1H-PHENANTHRO(9,10-D)IMIDAZOLES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-01-20 EP disclosed
EP-0043788-A1 Imidazole derivatives, process for their preparation and their pharmaceutical compositions SCHERING AKTIENGESELLSCHAFT (DE) 1982-01-13 EP disclosed
EP-0032113-A2 Antiinflammatory 4,5-diaryl-alpha-(polyhaloalkyl)-1H-imidazole-2-methanols E.I. DU PONT DE NEMOURS AND COMPANY (US) 1981-07-15 EP disclosed
US-4215135-A Antiinflammatory 2-substituted-1H-phenanthro[9,10-d]imidazoles E. I. DU PONT DE NEMOURS AND COMPANY (US) 1980-07-29 US disclosed
EP-0011115-A1 Antiinflammatory 2-substituted-1H-phenanthro(9,10-d)imidazoles, their preparation and pharmaceutical compositions containing them E.I. DU PONT DE NEMOURS AND COMPANY (US) 1980-05-28 EP disclosed
EP-0010361-A1 Bis-imidazoles, their preparation and pharmaceutical compositions containing them SMITHKLINE BECKMAN CORPORATION (US) 1980-04-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100184097-A1 4,5-BIS(4-METHOXYPHENYL)IMIDAZOLE COMPOUND INDUCING DIFFERENTIATION OF MYOBLASTS OR MUSCLE FIBERS INTO NEURON CELLS, A PHARMACEUTICAL COMPOSITION INCLUDING SAID COMPOUND, A METHOD OF INDUCING NEURON CELLS DIFFERENTIATION AND A SCREENING METHOD FOR IDENTIFYING ADDITIONAL COMPOUND USEFUL FOR INDUCING NEURON CELLS DIFFERENTIATION MUSK, TNNI3, TNNC1 MAPT 117/4885KDM4E 400/4885CYP3A4 99/4885
US-20050276764-A1 Topical use of bis-arylimidazo[1,2-a]thiolane derivatives ITCH, TRPA1, TPH1 MAPT 1423/4885KDM4E 1808/4885CYP3A4 1939/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.