SCHEMBL11265451

SCHEMBL11265451

O=C(c1ccccc1)c1c(Br)cc2n1CCC2C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC42 P60953 3/20 0.60
RAC1 P63000 3/20 0.60
PTGS2 P35354 3/20 0.60
PTGS1 P23219 2/20 0.60
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
CHRM3 P20309 1/20 0.60
OPRM1 P35372 1/20 0.60
PAK1 Q13153 1/20 0.60
HTT P42858 3/20 0.50
MAPK1 P28482 2/20 0.50
LMNA P02545 2/20 0.50
CYP1A2 P05177 2/20 0.50
ABCC4 O15439 1/20 0.50
BLM P54132 1/20 0.50
NFKB1 P19838 1/20 0.50
CA12 O43570 3/20 0.40
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
CA4 P22748 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11064934 0.90 CDC42 (0.49) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11271813 0.88 NPC1 (0.47) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL10935135 0.87 PTGS2 (0.47) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11270491 0.87 CDC42 (0.47) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11603510 0.86 CDC42 (0.60) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL10815779 0.86 CDC42 (0.45) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL10934380 0.85 CDC42 (0.59) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL10817308 0.85 CDC42 (0.44) CDC42RAC1PTGS2PTGS1NPC1
Hexane SCHEMBL11274049 0.84 CDC42 (0.45) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11272062 0.84 CDC42 (0.43) CDC42RAC1PTGS2PTGS1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4344943-A ANALGESICS, ANTIINFLAMMATORY AGENTS SYNTEX (U.S.A.) INC. (US) 1982-08-17 US claimed
EP-0041711-A1 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo(1,2-a)-pyrrole-1-carboxylic acids and derivatives thereof, process for their production and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1981-12-16 EP claimed
US-4344943-A ANALGESICS, ANTIINFLAMMATORY AGENTS SYNTEX (U.S.A.) INC. (US) 1982-08-17 US disclosed
EP-0041711-A1 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo(1,2-a)-pyrrole-1-carboxylic acids and derivatives thereof, process for their production and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1981-12-16 EP disclosed