SCHEMBL11270491

SCHEMBL11270491

O=C(c1cccc(F)c1)c1c(Br)cc2n1CCC2C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC42 P60953 3/20 0.47
RAC1 P63000 3/20 0.47
PTGS2 P35354 3/20 0.47
PTGS1 P23219 2/20 0.47
NPC1 O15118 1/20 0.47
CHRM3 P20309 1/20 0.47
OPRM1 P35372 1/20 0.47
RAB9A P51151 1/20 0.47
PAK1 Q13153 1/20 0.47
POLB P06746 1/20 0.41
HTT P42858 2/20 0.40
ABCC4 O15439 1/20 0.40
BLM P54132 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
NFKB1 P19838 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11265451 0.87 CDC42 (0.60) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11278560 0.87 CDC42 (0.46) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11271813 0.86 NPC1 (0.47) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11064934 0.81 CDC42 (0.49) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11357953 0.81 PTGS2 (0.74) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11602531 0.79 CDC42 (0.47) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11273207 0.77 CDC42 (0.45) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL10815779 0.77 CDC42 (0.45) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11269293 0.77 NPC1 (0.42) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11272575 0.77 CDC42 (0.42) CDC42RAC1PTGS2PTGS1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4344943-A ANALGESICS, ANTIINFLAMMATORY AGENTS SYNTEX (U.S.A.) INC. (US) 1982-08-17 US disclosed
EP-0041711-A1 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo(1,2-a)-pyrrole-1-carboxylic acids and derivatives thereof, process for their production and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1981-12-16 EP disclosed