SCHEMBL1126593

SCHEMBL1126593

CON(C)C(=O)C(Cc1ccccc1)N(C(=O)O)C(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.44
HPGD P15428 1/20 0.43
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
CTRB1 P17538 1/20 0.39
HTT P42858 2/20 0.38
MAPK1 P28482 1/20 0.38
ADAMTS5 Q9UNA0 1/20 0.38
LAP3 P28838 1/20 0.38
RIPK1 Q13546 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CHRM1 P11229 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP14 P50281 1/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21526204 1.00 FAAH (0.44) FAAHHPGDALDH1A1MAPTCTRB1
SCHEMBL8646560 0.90 FAAH (0.45) FAAH
SCHEMBL8647565 0.88 LDHA (0.48) FAAHALDH1A1HTTMAPK1MEN1
SCHEMBL9103138 0.87 KMT2A (0.41) FAAHHPGDALDH1A1CTRB1HTT
SCHEMBL28932692 0.86 HPGD (0.48) HPGDALDH1A1MAPTHTTADAMTS5
SCHEMBL2500069 0.86 HPGD (0.48) HPGDALDH1A1MAPTHTTADAMTS5
SCHEMBL8647911 0.83 ACACB (0.42) FAAHPPARGPPARA
SCHEMBL20524456 0.83 FAAH (0.48) FAAHHPGDALDH1A1MAPTHTT
SCHEMBL9329177 0.82 HPGD (0.50) FAAHHPGDALDH1A1MAPTHTT
SCHEMBL28656503 0.81 CYP1A2 (0.47) HPGDALDH1A1MAPTHTTADAMTS5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3788031-B1 DIPEPTIDYL KETOAMIDE META-METHOXYPHENYL DERIVATIVES AND USES THEREOF LANDSTEINER GENMED S L (ES) 2023-09-27 EP disclosed
US-11242312-B2 Dipeptidyl ketoamide meta-methoxyphenyl derivatives and uses thereof LANDSTEINER GENMED, S.L. (ES) 2022-02-08 US disclosed
US-20210317075-A1 DIPEPTIDYL KETOAMIDE META-METHOXYPHENYL DERIVATIVES AND USES THEREOF LANDSTEINER GENMED, S.L. (ES) 2021-10-14 US disclosed
EP-3564211-A1 DIPEPTIDYL KETOAMIDE META-METHOXYPHENYL DERIVATIVES AND USES THEREOF LANDSTEINER GENMED, S.L. (ES) 2019-11-06 EP disclosed
EP-2284178-A2 Inhibitors of cancer cell, T-cell and keratinocyte proliferation 4SC AG (DE) 2011-02-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11242312-B2 Dipeptidyl ketoamide meta-methoxyphenyl derivatives and uses thereof DPP4, DPP7, DPP3 FAAH 3147/4885HPGD 3507/4885ALDH1A1 1411/4885
US-20210317075-A1 DIPEPTIDYL KETOAMIDE META-METHOXYPHENYL DERIVATIVES AND USES THEREOF DPP4, DPP7, DPP3 FAAH 3147/4885HPGD 3507/4885ALDH1A1 1411/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.