SCHEMBL11265962

SCHEMBL11265962

N=C(NC(N)=O)Nc1ccc(I)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 2/20 0.45
SIGMAR1 Q99720 1/20 0.44
TRPV1 Q8NER1 3/20 0.44
IDO1 P14902 1/20 0.43
F2 P00734 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
TMPRSS6 Q8IU80 1/20 0.43
ST14 Q9Y5Y6 1/20 0.43
PEPD P12955 1/20 0.42
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
FPR2 P25090 3/20 0.39
EPHX1 P07099 1/20 0.39
EPHX2 P34913 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22939669 0.85 SIGMAR1 (0.47) CA12CA1CA2CA9SIGMAR1
SCHEMBL10735458 0.83 PEPD (0.64) CA12CA1CA2CA9F2
Hydrochloric Acid SCHEMBL9668364 0.83 SIGMAR1 (0.46) CA12CA1CA2CA9SIGMAR1
SCHEMBL4101986 0.81 ALDH1A1 (0.66) CA12CA1CA2CA9F2
SCHEMBL4100266 0.81 MEN1 (0.50) CA12CA1CA2CA9SIGMAR1
SCHEMBL4113103 0.81 NPC1 (0.66) CA12CA1CA2CA9F2
SCHEMBL2955430 0.81 GAA (0.55) F2PRSS1NPC1ALDH1A1EPHX1
SCHEMBL5533070 0.80 PEPD (0.64) CA12CA1CA2CA9SIGMAR1
Hydrochloric Acid SCHEMBL28052672 0.78 PEPD (0.61) CA12CA1CA2CA9SIGMAR1
SCHEMBL4105580 0.77 NPC1 (0.58) F2NPC1ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4115564-A Treatment of diarrhea with amidinoureas WILLIAM H. RORER, INC. (US) 1978-09-19 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed