SCHEMBL11267142

SCHEMBL11267142

CCC(=O)N1CCN(C(=O)OC2C3=C(SCC(OC)CS3)C(=O)N2c2ccc(Cl)cn2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.51
ADORA3 P0DMS8 1/20 0.51
MAPT P10636 1/20 0.51
RECQL P46063 1/20 0.51
GABRA1 P14867 1/20 0.51
GABRA3 P34903 1/20 0.51
GABRA2 P47869 1/20 0.51
GABRB2 P47870 1/20 0.51
GABRA4 P48169 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
NPSR1 Q6W5P4 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HRH3 Q9Y5N1 5/20 0.35
KDM4E B2RXH2 1/20 0.34
CHRM1 P11229 1/20 0.34
CKS1B P61024 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11266410 0.91 TSHR (0.63) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11268377 0.85 MAPT (0.35) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11846358 0.80 TSHR (0.53) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11263670 0.80 MAPT (0.42) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11833241 0.79 TSHR (0.65) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11277201 0.78 ADORA3 (0.47) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11829807 0.78 ADORA3 (0.54) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11260218 0.77 MAPT (0.39) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11847720 0.76 TSHR (0.52) TSHRADORA3MAPTRECQLGABRA1
SCHEMBL11263246 0.75 ADORA3 (0.44) TSHRADORA3MAPTRECQLGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4327095-A TRANQUICIZERS, ANTICONVULSANTS DECONTRACTURANTS AND HYPNOGENIC AGENTS RHONE-POULENC INDUSTRIES (FR) 1982-04-27 US claimed
US-4327095-A TRANQUICIZERS, ANTICONVULSANTS DECONTRACTURANTS AND HYPNOGENIC AGENTS RHONE-POULENC INDUSTRIES (FR) 1982-04-27 US disclosed